Thioctacid - capsules, mbadamba

Thioctacid BV: ntuziaka maka ojiji na nyocha

Aha Latin: Thioctacid

Koodu ATX: A16AX01

Ngwakọta ọrụ: thioctic acid (thioctic acid)

Onye na-emepụta: Nrụpụta GmbH MEDA (Germany)

Nkọwa na nwelite: 10.24.2018

Ego dị n'ụlọ ahịa ọgwụ: site na 1599 rubles.

Thioctacid BV bụ ọgwụ metabolic nwere mmetụta antioxidant.

Mwepụta wepụtara ya na ihe mebere

Thioctacid BV dị n'ụdị mbadamba ụrọ nwere ihe mkpuchi fim: akwụkwọ ndụ akwụkwọ ndụ-odo, obon biconvex (30, 60 ma ọ bụ 100. Na karama gbara ọchịchịrị, otu karama 1 na kaadiboodu).

Otu mbadamba 1 nwere:

  • ihe na-arụ ọrụ: thioctic (alfa-lipoic) acid - 0.6 g,
  • ihe inyeaka: magnesium stearate, hyprolose, hyprolose dị ala,
  • ihe mkpuchi ihe nkiri: titanium dioxide, macrogol 6000, hypromellose, aluminom varnish dabere na indigo carmine na dye quinoline odo, talc.

Omume ọgwụ

Coenzyme tinyere aka na oxarative decarboxylation nke pyruvic acid na alfa-keto acid na-arụ ọrụ dị mkpa na nguzo ike nke ahụ. Site na okike nke ihe ndu aru, lipoic acid yiri nke vitamin B. Ọ na-ekere òkè na nhazi nke lipid na carbohydrate metabolism, na-enwe mmetụta lipotropic, na-emetụta metabolism, na-eme ka ọrụ imeju, nwee mmetụta detoxifying ma ọ bụrụ na nsị na nnu ọla dị arọ na nsí ndị ọzọ.

Mmekorita

Ọgwụ a na - akwalite mmetụta mgbochi mkpali nke corticosteroids.

N'iji oge, a na-achọpụta mbelata nke arụmọrụ nke cisplatin. Ọgwụ ndị a na-ejikọ ọla, yabụ na ekwesighi ịkọ ha n'otu oge yana ọgwụ nwere ọla (dịka ọmụmaatụ, iron, magnesium, ngwaahịa nwere mmiri ara ehi nwere).

N'iji oge, a ga - eme ka ihe insulin na ọgwụ antidiabetic maka nchịkwa ọnụ, yabụ, a na-atụ aro ka ị na - agbaso ọkwa glucose ọbara mgbe ọ bụla, karịsịa na mmalite ọgwụ. N'ọnọdụ ụfọdụ, enwere ike belata ọgwụ nke hypoglycemic ọgwụ iji zere mmepe nke akara nke hypoglycemia (glucose ọbara dị ala).

Ọ bụrụ na ewere nkeji iri atọ tupu nri ụtụtụ, mgbe ahụ ị nwere ike ịme nkwadebe nwere iron ma ọ bụ magnesium n'ehihie ma ọ bụ na mgbede.

Mmanya na-egbu egbu nwere ike belata ịdị irè nke ọgwụ. Ya mere, a na-adụ ndị ọrịa ọdụ ka ha hapụ ị beụ ihe ọholicụholicụ na-egbu egbu n'oge a na-eji ọgwụ ahụ.

Mlọ ọgwụ

Thioctacid BV bụ ọgwụ metabolic na-eme ka neurons trophic dị elu, nwee ọrịa hepatoprotective, hypocholesterolemic, hypoglycemic, na mmetụta dị ala.

Ihe na-arụ ọrụ nke ọgwụ ahụ bụ thioctic acid, nke dị na ahụ mmadụ ma bụrụkwa antioxidant endogenous. Dịka coenzyme, ọ na-esonye na ọgwụ oxidative phosphorylation nke pyruvic acid na alfa-keto acids. Usoro ihe nke thioctic acid dị nso na mmetụta biochemical nke vitamin B Ọ na - enyere aka ichebe mkpụrụ ndụ site na nsonaazụ nsonaazụ nke radicals na - apụta na usoro metabolic, na - egbochi ihe ndị na - egbu egbu nke batara ahụ. Bawanye ọkwa nke antioxidant antioxidant glutathione, na-ebute mbelata ogo ihe mgbaàmà nke polyneuropathy.

Mmetụta mmekọrịta nke thioctic acid na insulin bụ mmụba nke itinye glucose.

Mlọ ọgwụ

Ntinye nke thioctic acid site na eriri afọ (GIT) mgbe ejiri ọnụ na-eme ya na-apụta ngwa ngwa na kpamkpam. Iji ọgwụ a were nri nwere ike belata mmịpụta ya. Cmax oke itinye uche na plasma ọbara mgbe ewerechara otu ihe na - enweta ya mgbe nkeji iri atọ ma ọ bụ 0.004 mg / ml. Ezigbo bioavailability nke Thioctacid BV bụ 20%.

Tupu abanye n'ọbara sistem, thioctic acid na-enwe mmetụta nke akụkụ nke mbụ gafere site na imeju. Mainzọ nke ụzọ nke metabolism ya bụ oxidation na conjugation.

Ndi1/2 (ọkara ndụ) bụ nkeji iri abụọ na ise.

Mwepu nke ihe na - arụ ọrụ bụ Thioctacid BV na metabolites ya na-arụ site na akụrụ. Site na mmamịrị, 80-90% nke ọgwụ na-adị.

Ntuziaka maka iji Thioctacid BV: usoro na usoro onunu ogwu

Dịka ntuziaka ahụ si dị, a na-ewere Thioctacid BV 600 mg n'ime afọ efu n'ime, awa 0,5 tupu nri ụtụtụ, na-elo ihe niile ma drinkingụọ nnukwu mmiri.

Usoro a tụrụ aro: 1 pc. Otu ugboro n'ụbọchị.

N'iburu ikike ogwu a, maka ọgwụgwọ nke ụdị polyneuropathy dị njọ, nchịkwa mbụ nke ihe ngwọta nke thioctic acid maka nchịkwa intravenous (Thioctacid 600 T) ga - ekwe omume maka oge nke ụbọchị iri na anọ ruo ụbọchị iri abụọ na asaa, nke a na - esote onye ọrịa na ị intụ ọgwụ kwa ụbọchị (Thioctacid BV).

Nsonaazụ

  • site na nri digestive: ọtụtụ mgbe - ọgbụgbọ, obere adịkarịghị - vomiting, mgbu afọ na eriri afọ, afọ ọsịsa, mebiri nke sensations
  • site na ụjọ usoro: oge ​​ụfọdụ - akpịrị,
  • mmeghachi omume nfụkasị ahụ: ọ dịkarịsịrị - itching, ọnya anụ ahụ, urticaria, urepula anafilactic,
  • site na anụ ahụ n'ozuzu ya: ọ dịkarịsịrị ike - mbelata ọbara glucose, ọdịdị nke ihe mgbaàmà hypoglycemia n'ụdị isi ọwụwa, ọgba aghara, ịba ụba ịba ụba, na nkwarụ anya.

Dodoụbiga ya ókè

Mgbaàmà: megide nzụlite otu uzu nke 10-40 g nke thioctic acid, mmerụ ahụ siri ike nwere ike ịmalite site na ngosipụta dịka njiri amamịghe juputara n'ọbara, hypoglycemic coma, nnukwu nsogbu na acid-base balance, lactic acidosis, nsogbu ọbara ọgbụgba siri ike (gụnyere ọnwụ).

Ọgwụ: ọ bụrụ na a na-enyo enyo enyo nke Thioctacid BV (otu mkpụrụ maka ndị okenye karia mbadamba 10, nwatakịrị karịrị 50 mg kwa 1 kilogram nke ahụ ya), onye ọrịa ahụ chọrọ ụlọ ọgwụ ozugbo yana nhọpụta nke usoro ọgwụgwọ Symptomatic. Ọ bụrụ na ọ dị mkpa, a na-eji usoro ọgwụgwọ anticonvulsant eme ihe, usoro mberede chọrọ iji nọgide na-arụ ọrụ nke akụkụ ahụ dị mkpa.

Ntụziaka pụrụ iche

Ebe ethanol bụ ihe dị egwu maka mmepe nke polyneuropathy ma na-ebute mbelata ọgwụgwọ Thioctacid BV, oriri mmanya na-egbochi ndị ọrịa.

Na ọgwụgwọ polyneuropathy na-arịa ọrịa shuga, onye ọrịa ahụ kwesịrị ịmepụta ọnọdụ ndị na-ahụ maka ịkwado ọkwa glucose dị n'ọbara.

Njirimara nke Thioctacid

N'ime ụlọ ahịa ọgwụ ị nwere ike ịzụta ngwaahịa a n'ụdị mbadamba BV (mwepụta ngwa ngwa) ma ọ bụ ngwọta. Iji hụ njimara nke kachasị mma na iwepu ọnwụ nke ihe, ngwa Ntọhapụ ngwa ngwa dabara adaba maka Njirimara nke thioctic acid. A na - ewepụta Acid ma na - etinye obi gị dum na afọ, mgbe ahụ, ozugbo a ga - amalite ịpụpụ. Mkpụrụ nke Thioctic acid anaghị agbakọ ma kpochapụrụ ya kpamkpam n'ahụ ahụ, ebe ọ na-etinye ego n'ọrụ na mweghachi na nchebe nke mkpụrụ ndụ.

A na - enweta Thioctacid n'ụdị mbadamba naanị maka ịhapụ ngwa ngwa, ebe ọ bụ na ụdị etinyere na-emetụta obere mkpirisi na enweghị atụ nke nsonaazụ ọgwụgwọ.

A na-ewere ọgwụ 1 mbadamba oge 1 kwa ụbọchị na afọ na-efu 20-30 nkeji tupu nri - n'oge ọ bụla n'ụbọchị. Enwere ike ịgwọta azịza ya na-enweghị dilution, mana a na-agbanye ya nnu na mmiri ma jiri nwayọọ nwayọọ, ọ bụghị ngwa ngwa karịa nkeji iri na abụọ, ya mere, a na-eme usoro a n'ụlọ ọgwụ.

Ihe kachasị dị n ’ọgwụ ahụ bụ ọgwụ alfa-lipoic (thioctic) n’ime ọnụọgụ 600 mg na mbadamba ọ bụla na ampoule nke ọ bụla.

Dịka akụrụngwa inyeaka, ihe ngwọta nwere trometamol na mmiri na-enweghị mmiri maka ntụtụ ma ọ nweghị ọgwụ etleyne acid, propylene glycols na macrogol.

Mbadamba ụrọ bụ ihe ndị dịkarịsịrị nta nke ọdịnaya, ejighi lactose, stachi, cellulose, mmanụ castor, nke a na-ahụkarị maka nkwadebe thioctic acid dị ọnụ ala.

Applicationzọ ntinye

Ihe dị na thiocic acid dị n'ọrụ na-ekere òkè na metabolism rụrụ na mitochondria - ihe owuwu nke mkpụrụ ndụ maka ịmalite nke ike ihe zuru ụwa ọnụ adenosine triphosphoric acid (ATP) abụba na abụba carbohydrates. ATP dị mkpa maka sel niile ịnata ike. Ọ bụrụ na ike ihe ezughị, yabụ sel agaghị enwe ike ịrụ ọrụ nke ọma. N'ihi ya, arụ ọrụ dị iche iche na arụ ọrụ akụkụ ahụ, anụ ahụ yana sistem nke akụkụ niile.

Thiocic acid bụ ọgwụ antioxidant dị egwu, nke dị nso na vitamin B n'ihe banyere usoro ya si arụ ọrụ.

Na ọrịa shuga mellitus, ị alcoholụbiga mmanya ókè na ọrịa ndị ọzọ, obere arịa ọbara na-abụkarị mkpọchi ma na-achịkwa nke ọma.

Eriri akwara, nke dị na oke anụ ahụ, na-enwe oke ụkọ nke nri dị mkpa yana ATP, nke na-ebute ọrịa. E gosiputara ha site na imebi ezi uche dị na ha na ebumnuche ụgbọ ala.

N'otu oge ahụ, ahụ erughị ala na mpaghara ahụ ebe akwara metụtara emetụta na-agafe. Ahụmahụ ndị na-adịghị mma gụnyere:

  • Ihe ọghọm nke sistem akụkụ ụjọ (ọnụọgụ, itching, inwe mmetụta na-ere ọkụ na nsọtụ, na -agagharị agagharị)
  • nsogbu nke sistem ara (eriri afọ dyskinesia, nsogbu nke akwara obi, dysfunction erectile, urinary incontinence, sweating, skin skin and other)

Iji kpochapụ ihe mgbaàmà ndị a, weghachite nri cellular, a chọrọ ọgwụ Thioctacid BV. Mkpụrụ ọgwụ a na-egbo mkpa nke mkpụrụ ndụ nke ọma maka eziokwu ahụ bụ na etolitela ATP zuru oke na mitochondria.

A na - ekepụta Thioctic acid n'onwe ya na mkpụrụ ndụ niile na - arụ ọrụ ọfụma n'ihi na achọrọ ya. Site na mbelata na ọnụọgụ ya, mmebi dị iche iche na-apụta.

Ọgwụ na-ewepụ adịghị ike nke ihe oriri yana mgbaàmà na-adịghị mma nke neuropathy mamịrị. Na mgbakwunye, a na-eji ọgwụ ahụ omume:

  1. antioxidant. Dịka antioxidant, ọ na - enyere aka ichebe sel nke sistem na akụkụ nke mmebi site na radicals n'efu, nke etolite n’oge mbibi ihe ndị si mba ọzọ na-abanye n’ahụ. Ọ nwere ike ịbụ ntụ ahụ, nnu nke ọla ndị dị arọ na nje virus,
  2. antitoxic. Ọgwụ na - enyere aka iwepu nhụsianya nke egbu egbu site na mkpochapu ngwa ngwa na mwepu nke ihe ndị na - emerụ ahụ,
  3. insulin-dị ka. Ọ dabere na ikike nke ọgwụ iji belata mkpokọ shuga n'ọbara site na ịbawanye uru site na mkpụrụ ndụ. N'ihi ya, ọgwụ ahụ na - eme ka ndị mmadụ nwee ike ịrịa ọrịa shuga, na-eme ka ahụike ha niile ma na - arụ ọrụ dịka insulin nke ha.
  4. na-atụnye ụtụ n’ibelata oke ibu (na-emeju agụụ, na-emebi abụba, na-eme ka ọrụ dum ka ọ dị mma ma na-adị mma),
  5. hepatoprotective
  6. ọrịa na-egbu egbu,
  7. ịbelata ike.

Ọ dị mkpa icheta na ọ dị mkpa ime ihe niile dọkịta depụtara maka ọgwụgwọ nke ọrịa na - akpata ọrịa shuga.

Ihe ngosi maka iji Thioctacid (BV)

Dịka anyị kwurula, a gosipụtara ọgwụ ahụ iji kpochapụ neuropathy na polyneuropathy na ị alcoholụ mmanya na mellitus shuga (nke nyocha nke ndị dọkịta na ndị ọrịa ha gosipụtara).

Ekwesịrị iburu mbadamba ihe ndị dị na Thioctacid minit 30 tupu nri. Is isụ ọgwụ kpamkpam. (Ọ naghị ata ata) ma jiri mmiri sachaa ya.

Ọ bụ dibia bekee ga-ekpebi oge ọgwụgwọ ọ bụla. Ike nke ọgwụgwọ ga-adabere:

  • ogo ọrịa ahụ,
  • ọnụego na mgbaàmà ya na-apụ n'anya
  • ọnọdụ onye ọrịa.

A na-atụ aro ogologo oge ọgwụgwọ, ebe ihe a bụ ihe dị maka anụ ahụ ma ọ naghị emeju. N'ezie, nke a bụ ọgwụgwọ mmechi. Ya mere, usoro dịkarịa ala bụ ọnwa 3 (enwere ngwugwu nke mbadamba 100, ihe kachasị echekwa ịzụta). Enwere nyocha nke nchịkwa na-aga n'ihu ruo afọ 4, nke gosipụtara nnwere onwe dị mma na nchekwa nke ọgwụ. Ọtụtụ ndị ọrịa na-ewere ya oge niile, ebe ọ bụ na emebi emebi ọrịa ahụ na akwara anụ ahụ na-echekwa ahụ ma ahụ ya chọrọ ihe a.

Site na oria bu oria di egwu, akwara ndi oria dika Thioctacid intravenly rue izu iri-abuo. Naanị mgbe mgbanwe a gachara iji Thioctacid rụọ ọrụ ogologo oge na 600 mg kwa ụbọchị.

Ojiji nke Thioctacid T

Ihe ngwọta nke ọgwụ Thioctacid T (600 mg) na usoro ahụike ka eji eme ihe maka nchịkwa intravenous kpọmkwem. Ihe ndị ahụ na-adọrọ adọrọ, yabụ ampoules gbara ọchịchịrị na agba, ekpuchiekwa karama ahụ nwere mmiri ga-eji kpuchie ya. Ọbara na-abanye n'ime nwayọ nwayọ. Dose 600 mg (1 ampoule) kwa ụbọchị. Dabere na ọgwụ dọkịta nyere, ọ ga-ekwe omume ịbawanye ọgwụ dabere n'ọnọdụ onye ọrịa.

Ọ bụrụ na ọrịa neuropathy na-arịa ọrịa shuga siri ike, mgbe ahụ a na-a drugụ ọgwụ ahụ maka izu abụọ na anọ.

N'ihe banyere mgbe onye ọrịa ahụ enweghị ike ịnata ụmụ irighiri Thioctacid 600 T n'ụlọ ọgwụ, ọ bụrụ na ọ dị mkpa, enwere ike dochie ha site na iji mbadamba Thioctacid BV na usoro ọgwụgwọ kwekọrọ, ebe ọ bụ na ha na-enye ọkwa zuru oke nke ihe ahụ na-arụ ọrụ n'ime ahụ.

Dabere n'ụkpụrụ ọgwụgwọ nke Ministry of Health nke Russian Federation, thioctic acid egosipụtara maka ịba ọcha n'anya, radiculopathies, wdg.

Iwu maka iwebata na ichekwa ọgwụ

Y’oburu na dọkịta debara mmanu di n’ime ya, yabụ onye obia kwesiri ịmara na aga-elebara ubochi niile anya n’otu oge. Ọ bụrụ na ọ dị mkpa, tinye 600 mg nke ihe ahụ kwesịrị ịgbanye nnu na mmiri (ị nwere ike ọbụna na obere obere). A na-eme nwayọ nwayọ nwayọ n'oge niile na-erughị 1.7 ml na 60 sekọnd - dabere na oke nke saline (a na-edozi saline 250 nkeji 30-40 iji zere hemostasis). Nyocha na-ekwu na usoro dị otú ahụ maka ndị ọrịa mamịrị bụ ezigbo.

Ọ bụrụ na achọrọ ya iji ọgwụ ahụ ọgwụ intravenously, mgbe ahụ na nke a, a na-ewere mkpịsị ugodi ahụ kpọmkwem site na ampoule n'ime sirinji ma nwee njikọ mgbapụta infusion na ya, nke na-enye ohere maka ọgwụ ntụtụ kachasị. Iwebata n’ime akwara gha di nwayọ ma o ghaghị nkeji iri na abụọ.

N'ihi eziokwu ahụ bụ na edozi edozi nke Thioctacid nwere mmetụta dị oke ọkụ na ìhè, a na-akwado ya ozugbo iji ya. A na-ewepụ ampoules na ihe ahụ naanị tupu ejiri ya. Iji gbochie mmetụta na-adịghị mma nke ìhè, a ga-eji nlezianya kpuchie akpa ahụ nwere ihe edozi.

Enwere ike idobe ya n'ụdị a karịa elekere 6 site na nkwadebe.

N'ihe banyere ịdoụbiga mmanya ókè na mmeghachi omume ọjọọ

Ọ bụrụ n ’ịdoụbiga ihe ókè emeela n’ihi ihe dị iche iche, yabụ ihe mgbapụta ya ga - abụ:

  • nsogbu nke ọgbụgbọ
  • gagging
  • isi ọwụwa.

Mgbe ị na-axụbiga mmanya oke, Thioxide BV gosipụtara site na nkụda mmụọ nke nsụhọ na ọgba aghara psychomotor. Mgbe ahu akwara acid na –eme ihe ahu na ahuhu ahuhu etolitela.

Ọgwụ ọgwụgwọ dị irè akọwapụtara anaghị adị. Ọ bụrụ na ị nwere ihe ọbụla na-enye gị nsogbu gbasara ịxụbiga mmanya ókè, ọ dị mkpa ịkpọtụrụ ụlọ ọrụ ahụike ozugbo o kwere omume maka usoro ọgwụgwọ ịgwọ ahụ iji mee ka ahụ kwụsị.

Mkparịta ụka ọgwụ ọjọọ

Iji n'otu oge eji Thioctacid BV:

  • cisplatin - na-agbada mmetụta ọgwụgwọ ya,
  • insulin, ọnya hypoglycemic na-elekọta mmadụ - nwere ike ịkwalite nsonaazụ ha, yabụ, achọrọ nlebara anya glucose ọbara dị larịị, ọkachasị na mmalite nke ọgwụgwọ njikọta, ọ bụrụ na ọ dị mkpa, a na-anabata mbelata ọgwụ nke hypoglycemic ọgwụ,
  • ethanol na metabolites ya - kpatara ike ịgwụ ọgwụ.

Ọ dị mkpa iburu n'uche ngwongwo nke thioctic acid na njikọta nke ọla mgbe ejikọtara ya na ọgwụ ndị nwere iron, magnesium na ọla ndị ọzọ. A na-atụ aro ka a nabata oriri nnabata ha n'ehihie.

Nyocha na Thioctacide BV

Nyocha nke Thioctacide BV na-enwekarị echiche ziri ezi. Ndị ọrịa nwere ọrịa shuga na-egosi mbelata ọbara shuga na ọkwa cholesterol, ahụike dị mma na ndabere nke iji ọgwụ ogologo oge. Otu akụkụ nke ọgwụ ahụ bụ mwepụta ngwa ngwa nke thioctic acid, nke na-enyere aka mee ka usoro metabolic dịkwuo elu ma wepụ ihe acid na-enweghị afọ ojuju, ntụgharị nke carbohydrates na ike.

E gosipụtara mmetụta ọgwụgwọ dị mma mgbe ị na-eji ọgwụ maka ọgwụgwọ nke imeju, ọrịa akwara, na oke ibu. N'iji ya tụnyere analogues, ndị ọrịa na-egosi ntakịrị ọnọdụ nke nsonaazụ achọghị.

N'ime ụfọdụ ndị ọrịa, ị takingụ ọgwụ ahụ enweghị mmetụta a tụrụ anya ya na iwelata cholesterol ma ọ bụ tinye aka na mmepe nke urticaria.

Ahapụ Gị Ikwu