Acekardol: ntuziaka maka ojiji, analogues na nyocha, ọnụahịa na ụlọ ahịa ọgwụ nke Russia
Ihe nọ n'ọrụ bụ acetylsalicylic acid. Ndabere nke usoro ihe eji eme ihe bu ihe nwere ike igbochi cyclooxygenase site na akụrụngwa na-arụ ọrụ, nke na-eme ka mgbochi nke mmepụta thromboxane A2 na mbelata agụkọta platelet. Mmetụta antiplatelet ahụ riri site na otu mbadamba ihe ruru otu izu.
Usoro ị doụ ọgwụ dị elu nwere ike inwe mmetụta ọgwụ na antipyretic (karịa 300 mg). Ọgwụ ahụ na-etinye obi gị dum na ngari nri ma ọ bụ naanị metabolized mgbe oge ịmịkọrọ.
Ihe ngosi maka iji Acecardol
Kedu ọgwụ ndị si?
Edere Acecardol maka angina na-akwụghị ụgwọ, iji gbochie ugboro ugboro iji gbochie nsogbu dị na myocardial, iji gbochie embolism ụkwara ume ọkụ (tinyere ngalaba ya) na mkpụrụokwu akwara dị omimi (ya na ịnọ ogologo oge, dịka ọmụmaatụ, n'oge ịwa ahụ ogologo oge).
Edere ọgwụ ahụ maka ndị ọrịa nwere ihe ndị dị ize ndụ (ịba ụba ahụ mmadụ, kọlesterol dị elu, ọrịa shuga mellitus, ụtaba, afọ, ọbara mgbali elu) iji gbochie nnukwu ọrịa myocardial infarction.
Ntụziaka maka iji Acecardol na-atụ aro ịgwọ ndị ọrịa ọgwụ mgbe mmerụ ahụ na arụ ọrụ vaskụla (wee mee, carotid angioplasty, endarterectomy nke akwara carotid, akwara akwara onagide grafting, arteriovenous shunting) iji gbochie thromboembolism.
Edere ọgwụ ahụ maka ndị ọrịa nwere ọgba aghara dị mkpirikpi nke inye ọbara n'ọbara iji gbochie ọrịa azụ mgbu.
Ihe ngbanwe
Echighi ọgwụ a nye ndị ọrịa nwere ọrịa mbuze na ọnya akwara nke digestive, yana hemorrhagic diathesisọbara ọgbụgba site na afọ, duodenum. Edeghị ọgwụ a maka ụkwara ume ọkụ bronchial site na ị salụ salicylates.
A na-egbochi ọgwụ a na ọrịa ọrịa imeju obi obara, ya na usoro ọmụmụ nke sistem gbasara akụrụ, ebe a na-enye nwa ara.
Agbanyeghị oge ịgwọ ọrịa ọgwụ na methotrexate na usoro onunu ogwu kariri 15 mg kwa izu.
Ojiji Acecardol nwere oke na ndị ọrịa nwere hyperuricemia, gout, allergies ọgwụ, fever fever, nasals polyposis.
Acetylsalicylic acid nwere ike ibute ọbara ọgbụgba n'oge ịwa ahụ.
Nsonaazụ
Ọna nri: mmụba nke ALT na enzymes AST, vomiting, obi mgbawa, ọgbụgbọ, ọnya afọ, na ọbara ọgbụgba.
Usoro nke Hematopoietic: anaemiaihe egwu ọbara ọgbụgba n'ihi mgbochi nke nchịkọta platelet.
Azịza Allergic n'ụdị ọrịa obi, nfuchi nke azụ mucous nke imi imi, rhinitis, urticaria, ọnya Quincke, itching na ihe ọkụ ọkụ. Mmeghachi omume nfụkasị ahụ nke ụdị ahụ adịkarịghị amalite. anafilaisis.
Usoro okuku ume: spasm nke ọla aka nke obere ma di omimi.
Usoro ụjọ: ọhụhụ ụzọ nhụjuanya, tinnitus, isi ọwụwa, ọgbụgbọ.
Ngwakọta na ụdị ntọhapụ
Acecardol dị n'ụdị mbadamba ụrọ, bụ nke a na-eji mkpuchi na-adịghị mma, na 50, 100 na 300 mg. Mbadamba ọgwụ ahụ biconvex na okirikiri, na-acha ọcha (ikekwe ọ fọrọ nke nta ka ọ bụrụ ọcha) na agba. A na-ere ha na paịlị mbadamba 10. Otu kaadiboodu nwere ngwugwu ato.
- Ihe kachasị na-arụ ọrụ na Acecardol bụ acetylsalicylic acid.
- Ihe ndi ozo Acecardol bu: povidone di omimi, oka di na ala, lactose monohydrate, magnesium stearate.
Linlọ ọgwụ na ọgwụ ọgwụ: NSAIDs. Onye na-ahụ maka ihe mgbochi.
Ngwongwo ogwu
Ihe na-arụ ọrụ bụ acetylsalicylic acid. Ndabere nke usoro ihe eji eme ihe bu ihe nwere ike igbochi cyclooxygenase site na akụrụngwa na-arụ ọrụ, nke na-eme ka mgbochi nke mmepụta thromboxane A2 na mbelata agụkọta platelet. Mmetụta antiplatelet ahụ riri site na otu mbadamba ihe ruru otu izu.
Usoro ị doụ ọgwụ dị elu nwere ike inwe mmetụta ọgwụ na antipyretic (karịa 300 mg). Ọgwụ ahụ na-etinye obi gị dum na ngari nri ma ọ bụ naanị metabolized mgbe oge ịmịkọrọ.
Ntụziaka maka ojiji
Dabere na ntuziaka maka ojiji, a na-ewere Acecardol ọnụ tupu nri, yana nnukwu mmiri. O bu n'uche ogwu a ka o jiri ogologo oge.
- Mgbochi nke ọrịa myocardial na-enyo enyo: 100 mg / ụbọchị kwa ụbọchị ma ọ bụ 300 mg kwa ụbọchị ọ bụla (a ga-ata ata mbadamba mbụ maka nnabata ngwa ngwa).
- Mgbochi nke mbụ myocardial infarction na ọnụnọ ihe ndị dị ize ndụ: 100 mg / ụbọchị kwa ụbọchị ma ọ bụ 300 mg kwa ụbọchị.
- Mgbochi nke thromboembolism mgbe ịwa ahụ na mgbochi vaskụla mmerụ ahụ: 100-300 mg / ụbọchị kwa ụbọchị.
- Mgbochi ọnya afọ ischemic na ọrịa ụbụrụ nke na-efe efe: 100-300 mg / ụbọchị kwa ụbọchị.
- Mgbochi nke thrombosis nke miri emi na thromboembolism nke akwara ọbara na alaka ya: 100 mg / ụbọchị ma ọ bụ 300 mg kwa ụbọchị.
- Mgbochi nke infarction myocardial ugboro ugboro na angina na-akwụghị chịm: 100-300 mg / ụbọchị kwa ụbọchị.
N'oge usoro ọgwụgwọ yana nkwadebe dabere na acetylsalicylic acid, a ga-enyocha ule ọbara kwa oge, ebe ihe a na - enye aka na ịmịcha ọbara ya. Site na iji kaadi kaadi ogologo oge na enweghị nchịkwa, ihe ọghọm nke ịmalite ọbara ọgbụgba n'ime ahụ dị oke.
Hụrụ onye iro a swornụrụ iyi MUSHROOM nke mbọ! A ga-asacha mbọ gị na ụbọchị 3! Were ya. | |
Kedu otu esi eme ka nrụgide olu ike ngwa ngwa mgbe afọ 40 gasịrị? Ntụziaka ahụ dị mfe, dee ya. | |
Ike gwụrụ ọbara? E nwere ụzọ mgbapụ! Enwere ike ịgwọ ya n’ụlọ n’ụlọ ụbọchị ole na ole, ịkwesịrị. | |
Banyere ọnụnọ ikpuru na-ekwu ODOR site n'ọnụ ya! Otu ugboro n'ụbọchị, aụọ mmiri nwere mmiri iji .. NsonaazụDika nyocha, Acecardol na analog ya nwere ike ibute nsogbu ndi a:
O yikarịrị ka ịdoụbiga ihe ókè na-arụ ọrụ, ebe ọ bụ na ihe na-arụ ọrụ, acetylsalicylic acid, dị na obere ego. Cessụbiga ASA oke ókè nwere ike ibute ọbara ọgbụgba. Ime na lactationGgba ime na ịrara bụ ihe ndị ọzọ na - egbochi ọgwụ ọgwụ Acekardol. Amachibidoro ihe mgbochi mgbochi dị na mkpụrụ ụbọchị nke atọ na nke atọ nke afọ ime, na nke abụọ n’ime ọnwa nke abụọ ka ọ ga-akpachara anya ma bụrụkwa naanị onye dọkịta gwara ya. Ntinye na oge nke ọnwa nke abụọ bụ naanị ihe dị mma ga-enyere gị aka ma ọ bụrụ na ọ ga-abara nne ma ọ bụ nna ya aka karịa ihe o nwere ike ime. Analogs AcekardolAnakpụrụ nke analogues nke na-arụ ọrụ:
Ntị: iji ọgwụ ike ana-ekwenye ekwenye na dọkịta na-ahụ maka ịga. Ọnụ ego nke ATSECARDOL, mbadamba ihe dị na ụlọ ahịa ọgwụ (Moscow) bụ 25 rubles. Mwepụta wepụtara ya na ihe mejupụtaraA na-emepụta Acecardol n'ụdị mbadamba biconvex gburugburu, nke a na-etinye na shei ọcha. Otu mbadamba 1 nwere:
NsonaazụNtụziaka ahụ dọrọ aka ná ntị banyere ihe ga-ekwe omume ịzụlite mmetụta ndị a na-esochi mgbe ị na-ede akwụkwọ Acekardol:
Ihe ngbanwe Acekardol na contraindicated na ndị a:
Nyefee ya na nlezianya mgbe:
Dodoụbiga ya ókè Symptoms symptomsụbiga ihe ọdoụ includeụ ókè gụnyere ọgbụgbọ, ọgbụgbọ, isi ọwụwa, ọgba aghara, tinnitus, ịsụsọ oke, tachypnea, na hyperventilation. Na-atụ aro lavage gastric, iji carbon na-arụ ọrụ na mweghachi nke nguzo mmiri-electrolyte. Site na ịdoụbiga mmanya ókè, enwere ike - ahụ ọkụ dị oke elu, nsogbu iku ume, akwara obi, usoro ụjọ, glucose metabolism, na-agba ọbara na afọ na eriri afọ. N'okwu a, ụlọ ọgwụ ngwa ngwa na ọgwụgwọ mberede, gụnyere ịsacha eriri afọ, iji carbon ugboro ugboro, akụrụngwa ịwa ahụ, nrụgide alkaline diuresis, mweghachi nke acid-base steeti na mmiri-electrolyte, yana nhọpụta ọgwụgwọ symptomatic iji wee kpochapụ usoro mmepe. imebi. Ntụziaka pụrụ icheAcekardol nwere ike kpalite nkụchi obi na ọrịa ashma. Ihe ndị dị ize ndụ: akụkọ ihe mere eme nke polyposis nke imi, fever fever, allergy ọgwụ, ụkwara ume ọkụ. Mmetụta dị na igbochi nchịkọta platelet na-adịgide ruo ọtụtụ ụbọchị, nke nwere ike ibute ọbara ọgbụgba n'oge ọrụ ịwa ahụ mberede. Tupu ịmalite ọrụ, ịkagbu ọgwụ ahụ ọbụlagodi 7 ụbọchị tupu. N'ime ndị ọrịa nwere nsogbu, Acecardol na obere doses nwere ike ibute gout. N'ihe dị ize ndụ bụ ndị nwere ntakịrị uric acid excretion. Site na mmụba nke ọgwụ ahụ, ohere ịba ọbara ọgbụgba na-abawanye nke ukwuu. Ọ naghị emetụta ike ịnya ụgbọ ala. Na ọgwụgwọ nke glucocorticosteroids, a gharịrị iburu n'uche na site na kagbuo ha, enwere ike ịdoụbiga mmanya ókè. MmekoritaIhe oriri Acecardol na-akwalite nsị nke methotrexate, na-ebelata mwepụ akụrụ ya, valproic acid. Na-eme ka mmetụta nke NSAID ndị ọzọ, narcotic analgesics, ọgwụ ọgwụ hypoglycemic, heparin, anticoagulants na-apụtaghị ìhè, thrombolytics na ndị nnọchi antiplatelet, sulfonamides (gụnyere co-trimoxazole), T3. Na-ebelata mmetụta ọgwụ ọgwụ uricosuric (benzbromarone, sulfinpyrazone), ọgwụ antihypertensive, diuretics (spironolactone, furosemide). Ọgwụ GCS, ethanol na ethanol nwere ọgwụ na-abawanye mmetụta na-emebi emebi na mucosa, na-abawanye ohere nke ọbara ọgbụgba. Na-eme ka mkpokọ digoxin, barbiturates, na Li + nke dị na plasma na-abawanye ụba. Ihe antacids nwere Mg2 + na / ma ọ bụ Al3 + na-akwụsịlata ma gbochie mmịpụta nke ASA. Ọgwụ Myelotoxic na-eme ka ngosipụta nke ọgwụ ọgwụ ọgwụ dịkwuo elu. Acecardol, ntuziaka maka ojiji (Usoro na usoro onunu ogwu)A na-atụ aro ị medicineụ ọgwụ a tupu nri. Ọ bụ ihe amamihe dị na ị toụ mbadamba mmiri nwere oke mmiri mmiri. Edere ọgwụ a ogologo oge. Otutu maka ntinye - oge 1 kwa ụbọchị. Ọ bụrụ na eche na infarction myocardial siri ike maka mgbochi họpụta 100 mg kwa ụbọchị ma ọ bụ 300 mg kwa ụbọchị. Mbadamba mkpụrụ osisi na-ata ata, ọ na-eweta nsonaazụ ọsọ ọsọ, nke dị ezigbo mkpa na awa mbụ nke infarction myocardial. Ọ bụrụ na enwere ọtụtụ ihe ọghọm n'otu oge, 300 mg kwa ụbọchị, ma ọ bụ 100 mg kwa ụbọchị, ka edepụtara maka mgbochi nke nnukwu myocardial infarction. Mgbochi nke angina pectoris ejighị n'aka, nkụchi obi ugboro ugboro, mgbochi nke ọrịa ụkwara ume ọkụ, afọ ischemic: 100-300 mg kwa ụbọchị. Maka mgbochi nke ụkwara ume ọkụ, akwara nke nwere ume ala họta 300 mg kwa ụbọchị, ma ọ bụ 100 mg kwa ụbọchị. Dodoụbiga ya ókèMgbaàmà dị nwayọ dịka ọgbụgbọ, ọgbụgbọ, isi ọwụwa, ọgba aghara, tinnitus, ịsụsọ oke, tachypnea, na hyperventilation ga-ekwe omume. N'okwu a, ọgwụgwọ ahụ ga-etinye oke ndụ gastric, oriri dị elu nke carbon na-arụ ọrụ, na iweghachi nguzo mmiri-electrolyte. N’oké njọ nke ịdoụbiga mmanya ókè, ga-ekwe omume: ahụ ọ̀tụ̀tụ̀ ahụ dị elu, nsogbu iku ume, usoro akwara obi, sistem, glucose metabolism, na-agba mmee afọ na eriri afọ. N’okwu a ọ dịkwa mkpa ịnweta ụlọ ọgwụ ngwa ngwa. Mlọ ọgwụMgbe nchịkwa ọnụ gachara, ASA na-aracha ngwa ngwa kpamkpam na eriri afọ, n'oge a na-emegharị ya obere. N'oge oriri na mgbe a gbasachara, ASA na-agbanwe n'ime metabolite bụ isi - salicylic acid, nke metabolized kachasị na imeju (n'okpuru enzymes) iji mepụta metabolites dịka salicylic acid, salicylic acid glucuronide na phenyl salicylate. A na-ahụta ha n'ọtụtụ akwara na mmamịrị. N'ime ụmụ nwanyị, usoro metabolic dị nwayọ karịa na ụmụ nwoke. Mgbe ị gachara Acecardol n'ime, a na-ahụta ịta kachasị nke ASA na plasma ọbara mgbe nkeji 10-20 gasịrị, salicylic acid - mgbe awa 0.3-2 gasịrị. A na-eji mbadamba Acecardol mee ihe na-egbochi acid, nke na-egbochi ọgwụ ịgwakọta na afọ, yabụ ewepụtara ihe dị n'ọrụ na gburugburu alkaline nke duodenum. N'akụkụ a, nnabata nke ASA bụ awa 3-6 dị ala karịa mgbe ị na-ewere mbadamba ụrọ (ọ bụghị ihe mkpuchi dị ka shei). Acetylsalicylic na salicylic acid na-ekekọta protein ndị dị na plasma (ọ dabere na dose ahụ, ihe ngosi a bụ 66-99%) ma keere ya ngwa ngwa. Acid Salicylic na-aga n’iru Plasenta na n’ime mmiri ara. A na - egbochi metabolism nke salicylic acid site n'ike nke sistemụ enzymatic, yabụ, ntụpọ ya bụ nke dabere na ya.Ọkara ndụ ahụ na-adị site na awa 2-3 (n'ihe banyere obere doses) ruo awa iri na ise (mgbe ị na-eji ọgwụ ndị dị elu dị ka ọgwụ nje na ọgwụ). Site n'iji ogologo oge, ASA na-enweghị mmiri adịghị agbakọ n'ọbara ọbara, n'adịghị ka salicylates ndị ọzọ. Salicylic acid na metabolites ya bụ akụrụ. Site n'ịrụ ọrụ akụrụ dị, site na 80 ruo 100% nke otu ASA na-apụ apụ n'ime awa 24-72. Usoro onunu ogwu na nhaziA na-ewere mbadamba Acecardol tupu nri, were mmiri sachaa ya. O bu n'uche ogwu a ka o jiri ogologo oge. Ọ bụrụ na enyo infarction myocardial, a na-ewere Acecardol 100 mg otu ugboro n'ụbọchị ma ọ bụ 300 mg kwa ụbọchị. Maka mmetụta ọgwụgwọ kachasị mma, enwere ike ịta ụrọ nke mbụ. Iji gbochie infarction myocardial ugboro ugboro, ịchikọta akwara mkpụrụ osisi na akwara ya na mkpụkọ ọbara, verom thrombosis nke miri emi ma nwee angina na - ejighi ike, a na - ewere Acecardol 100-300 mg kwa ụbọchị. Iji gbochie thromboembolism mgbe mmerụ ahụ na usoro ịwa ahụ, usoro ọgwụgwọ Acecardol bụ 100-300 mg kwa ụbọchị. Ime na lactationN’ime oge izizi nke ịtụrụ ime, a na -eme ka ihe eji ebunye ya oke n’ọrụ iji mepụta ntụpọ n’ime nwa ebu n’uka (kea ugwu, ntụpọ obi), ya mere Acecardol machiri ihe eji eme ya. N’ime oge nke abụọ nke ịtụrụ ime, a ga - edenye ọgwụ ahụ naanị ma ọ bụrụ na uru a tụrụ anya ga - adị elu karịa ihe ọghọm ọ bụla. N'otu oge ahụ, a na-atụ aro iji Acecardol na usoro onyonye ihe na-erughị 150 mg maka usoro kachasị mkpụmkpụ. N'ime oge nke atọ nke afọ ime, salicylates na nnukwu onyonyo (karịa 300 mg / ụbọchị) na-ebelata ọrụ, na-ebute oke ọbara na nne na nwa ebu n’afọ, na mmechi oge akwara mkpụrụ ndụ nọ n’ime nwa ebu n’afọ. Iburu ASA ozugbo amụrụ nwa nwere ike ibute ọbara ọgbụgba n'ime intracranial, ọkachasị na ụmụ aka. N'akụkụ a, n'oge ọnwa ikpeazụ nke afọ ime, Acecardol machibidoro contraindicated maka iji ya. Salicylates na metabolites ha na-abanye n’ime mmiri ara, nke mere na a na-egbochi Acecardol n’ime ụmụ nwanyị na-enye nwa ara. Ọ bụrụ n ’ị theụ ọgwụ ziri ezi n’etiti ụlọ ọgwụ, ị kwesịrị ịkwụsị inye ara. Mkparịta ụka ọgwụ ọjọọN'ihe banyere iji otu oge, acetylsalicylic acid na-ebelata ike nke ọgwụ ndị a: diuretics, angiotensin-converting enhibme inhibitors (ACE), uricosuric ọgwụ (benzbromarone). N'ihe banyere iji otu oge, acetylsalicylic acid na-eme ka ihe omume nke ọgwụ ndị na-esonụ pụta: ndị na-egbochi antiplatelet na ọgwụ thrombolytic, digoxin, heparin na anticoagulants na-apụtachaghị ìhè, methotrexate, valproic acid, hypoglycemic ọgwụ (insulin na sulfonylurea n'ụdị). Ọzọkwa, njikọta nke ASA na methotrexate bụ ihe metụtara ọghọm nke mmeghachi omume akwara site na akụkụ ahụ haemopoietic, yana thrombolytics, ndị nnọchi ọgwụ antiraplet na ọgwụ anticoagulants - ohere dị elu nke ọbara ọgbụgba. ASA na - akwalite nsị na ethanol na sistemụ akwara. Nke a na - enye ohere nke mmebi ahụ ga-eme ka eriri afọ na oke ọbara na-anọ ogologo oge. Usoro glucocorticosteroids na-eme ka ikpochapụ ọgwụ kwụsị, karịa iweda mmetụta ya ike. Ihe analogues nke Acecardol bu njikere Thrombo ACC, Aspirin, Cardiopyrine, Aspinate, Aspicor, Taspir, Thrombopol, Acetylsalicylic acid. Nyocha na AcecardolDabere na nyocha, Acekardol bụ onye na - arụ ọrụ antiplatelet nke na - egbochi ọbara ma na - egbochi thrombosis. Uru ya ndị ọzọ gụnyere ọnụahịa dị ala (ma e jiri ya tụnyere ọtụtụ analogues), ịdị mfe nke nchịkwa (oge 1 kwa ụbọchị), ụdị usoro onunu ogwu (mkpuchi ihe na-echebe afọ na mmetụta ọjọọ nke acetylsalicylic acid), yana ọnụnọ nke usoro dị iche iche nke mbadamba (50, 100 na 300 mg), nke na-enye gị ohere ịhọrọ nke kachasị mma. Ọdịmma nke Acecardol gụnyere ọnụnọ nke contraindications. Agbanyeghị, ha dị maka salilylates niile, yabụ dọkịta kwesịrị ịkọwa ọgwụgwọ. |