Atoris mbadamba nkume analogues

N'iji Atoris (ma ọ bụ analogues), enwere ike nweta nsonaazụ dị mma na ọgwụgwọ hyperlipidemia na ọrịa obi. A na-eji ọgwụ ọzọ eme ihe iji gbochie ọnọdụ ndị a na ndị gafere afọ 55. Atoris rụpụtara ezigbo ọrụ, yabụ ịkwesịrị ịtụle atụmatụ nke iji ya, yana nkọwapụta nke mkpụrụ ego ndị na-adịghị ọnụ. Ndị a gụnyere ọgwụ ọjọọ dịka Lipoford, Atomax, na Atorvastatin. Ihe edere edere nke ogwu ahu na Atoris n’onwe ya nwere ihe ha na eme bu mmanu ndi emebere aru - caline atorvastatin.

Nkọwa nke Atoris

Mpempe akwụkwọ Atoris dị na ngwugwu nwere usoro ọgwụ nke 10, 20, 30, 40, 60 ma ọ bụ 80 mg. Nke a bụ ọgwụ statin na-arụ ọrụ ụfọdụ. Calcium Atorvastatin na-enyere aka belata ọrụ nke enzyme, nke bụ ihe na-enyere aka maka ntụgharị nke HMG-CoA na mevalonic acid. Mwepu nke mgbanwe a na-egbochi irighiri cholesterol, na-ewepụ ha na arịa. Nke a na-ebelata ihie LDL cholesterol n'ime ọbara.

Mbadamba mkpụrụ ndụ Atoris nwere mmetụta anti-atherosclerotic, nke na-egosipụta onwe ya site na ọrụ nke ihe bụ isi na arịa ọbara na akụkụ ọbara.

Mmetụta ziri ezi nke atorvastatin n’elu akwara ọbara dị n’aka na-egbochi ikerechi isoprenoids, nke na-ebelata ohere ịba ụba nke oghere dị n’ime ha, nke pụtara mbelata oghere ha.

N'etiti usoro izugbe maka ị theụ ọgwụ, enwere ike ịmata ọdịiche ndị a:

  1. Adrapagidesi ike na nri (tupu yana n'oge ọgwụgwọ) ga - enyere aka belata egbugbere ọnụ ọbara.
  2. Ekwesịrị ị drugụ ọgwụ ahụ n'otu oge 1 otu oge kwa ụbọchị.
  3. Ọ dị mkpa ịdị na-enyocha mgbe niile ihe ndị na-egosi ọrụ imeju.
  4. Site na mmepe nke mgbu akwara ma ọ bụ adịghị ike nke ọdịdị amaghi, tinyere ahụ ọkụ, a na-atụ aro ịkwụsị ịhapụ Atoris ma kpọtụrụ dọkịta.
  5. Atoris bụ contraindicated na ụmụntakịrị, yana ụmụ nwanyị n'oge a na-enye nwa ara na ime ime.
  6. Otu n'ime contraindications bụ ọdịda nke imeju, ọrịa imeju, akwara ọkpụkpụ.
  7. Ọ bụrụ na enwere otu akụkụ nke ọgwụ ahụ, na-adịghị akwado ọgwụ nchịkwa ya.
  8. Extremekpachapụ anya kwesiri ka e mee ndị ọrịa na-ahoụbiga mmanya ókè aka.

Mgbe izu 2 gachara ọgwụgwọ, cholesterol ọbara ga-ada. Nke a ga - apụta na nyocha. Enwere ike inwe mmetụta kachasị elu mgbe ụbọchị 25-30 gasịrị. Ọgwụgwọ ọgwụgwọ sitere na ọgwụgwọ ga-adịgide karịa naanị mgbe ịmechara usoro dọkịta niile nyere. N'okwu a, usoro ọgwụgwọ ahụ ka a ga-ekpebi ọkwa mbu nke LDL kọlesterol dị n'ọbara yana ogo ọrịa ahụ.

Njirimara nke iji ọgwụ analog Lipoford

Lipoford sitere na ndi India ma bu okwu Atoris di onu ala. Ọgwụ dị n'ụdị mbadamba nkume nwere mkpokọta akụkụ akụrụngwa nọ n'ọrụ 10 ma ọ bụ 20 mg. Lipoford bụ ọgwụ dị ala nke belata nke a na-eji na mgbochi na ọgwụgwọ nke ọrịa obi kpatara oke cholesterol.

Ihe banyere Lipoford na Atoris bụ ihe fọrọ nke nta ka ọ bụrụ otu, ebe ha abụọ gụnyere calcium atorvastatin dị ka isi ihe na-arụ ọrụ. Ma iji dochie anya Atoris na ọnụọgụ dị ọnụ ala, ọ dị mkpa ịkpọtụrụ dọkịta nke nyere ọgwụgwọ ahụ.

Ihe ngosi maka iji Lipoford nwere ike ịbụ otu n'ime ọnọdụ:

  • ịba ụba nke cholesterol,
  • mụbara LDL cholesterol
  • ọbara mgbali elu nke apolipoprotein B na triglycerides,
  • isi, heterozygous ezinụlọ na hypercholesterolemia na-abụghị nke ezinụlọ (ma ọ bụrụ na LDL cholesterol dị oke),
  • homozygous familial hypercholesterolemia,
  • gwakọtara na hyperlipidemia,
  • nnukwu ọnya triglyceride,
  • dysbetalipoproteinemia,
  • pathology nke obi usoro,
  • ihe egwu nke ibute ọrịa obi: ịka nká, nicotine riri ahụ, ọrịa shuga, wdg.

Mgbe ị na-eji Lipoford, ịkwesịrị ịgbaso nri pụrụ iche. Ihe oriri kwesịrị isi na nri cholesterol dị ala.

Atomax bu ihe omumu ozo nke Atoris

Atomax bu onye Atoris ndi India nke ozo jiri onu ahia kari ahia. Thedị mgbapụta ahụ bụ otu. Mbadamba ụnụ dị naanị n ’ụzọ abụọ: 10 na 20 mg. Akụkụ bụ isi nke Atomax bụ atorvastatin calcium trihydrate. Ihe mejupụtara ya gụnyere ihe dị ka ngwa iri ọzọ, gụnyere lactose, crospovidone, stachi, wdg.

A na-eji ọnụọgụ Atomax ọnụ, n'agbanyeghị nri ahụ. A na-etinye ọgwụ ahụ nke ọma, mgbe awa 1-2 gasịrị, a na-ahụta ntinye uche nke kachasị arụ ọrụ n'ime ọbara.

Ihe ndi choro ime ka oria Atomax nwere ike bu:

  • nfụkasị nke ihe mejupụtara ngwaahịa ahụ,
  • ime n’oge ọ bụla
  • inye ara
  • mmebi nke ọrịa imeju,
  • ụba ọrụ ọbara transaminase,
  • afọ ụmụaka
  • alisụrụma
  • ọrịa ọrịa imeju ọ bụla (jiri ngwaahịa na-akpachara anya ma na-elekọta dọkịta mgbe niile),
  • nsogbu electrolyte,
  • nsogbu na usoro endocrine,
  • mmebi nke usoro nje (dịka ọmụmaatụ, sepsis),
  • ọrụ ịwa ahụ, wdg.

Isi ihe onye ọrịa ahụ kwesịrị icheta: Enwere ike iji Atomax nwere cholesterol mee ya, kama ọ bụ naanị dị ka dọkịta si kwuo. Nke a bụ n'ihi n'eziokwu na site na iji ọgwụ na-adịghị mma, enwere ike ịme ka ụdị mmetụta dị iche iche na-abawanye ọtụtụ oge.

Onye na-anọchi anya Atorvastatin

N'etiti ọgwụ ụlọ nwere ike dochie Atoris, ekenyela ọgwụ nke nwere aha na isi ya - Atorvastatin. Ọ na-akwụ ụgwọ dị ala karịa analogues nke Atoris niile, dịka a na-emepụta ya na Russian Federation ma ọ bụghị ná mba ofesi. Ma n'ihe banyere ịdị irè, ọgwụ adịghị njọ. A na-emepụta mbadamba dị iche iche n'ọtụtụ ihe ike: 10-40 mg.

Enwere ike inye ogwu a maka otu ihe ngosi a ka ogwu ndia di n’elu, ebe obu na ihe ha n’otu dika ihe ndi ozo. N'ime ihe ndị kachasị na contraindications bụ ịtụrụ ime, inye ara, ọrịa imeju na nnukwu ọnọdụ, na ntachi obi mmadụ.

Otu nsogbu ndị a pụrụ inwe pụrụ ịpụta:

  • nsogbu ụra
  • isi ọwụwa
  • imebi akwa (afọ ọsịsa, afọ ntachi),
  • ọgbụgbọ
  • ịmụba ikuku n'ime eriri afọ,
  • izugbe oria
  • azu mgbu
  • ogwe
  • akpukpo aru, wdg.

Ọ bụrụ na cholesterol dị elu, akụrụngwa ga - enyere aka ịnagide nsogbu ahụ, mana ọ dabere na usoro kwesịrị ekwesị. Ya mere, ọ dị ezigbo mkpa ịrapagidesi ike na usoro ọgwụgwọ dọkịta depụtara. N'ihe banyere ịdoụbiga mmanya ókè, a kwụsịrị ị drugụ ọgwụ ahụ. Enwere ike igbochi mmịcha ọzọ site na ịsacha afọ, na-egbu mgbu ma ọ bụ ụfọdụ ihe na-anabata ihe. Na mgbakwunye, dọkịta ahụ nwere ike ịkọwa ọgwụgwọ Symptomatic, nke a ga-elekwasị anya na nyochaa ma nọgide na-arụ ọrụ ndị dị mkpa.

Ihe oriri Atoris dị ọnụ ala

Ihe analogue dị ọnụ ala site na 250 rubles.

Emere dochie anya nke a na Russia, yabụ ọ na-efu ihe na-erughị "ọgwụ mbụ". O nwere otu uzo ihe ngosi banyere oge a. Contraindicated bụrụ na hypersensitivity na ọgwụ, ọrịa imeju, n'oge ime na lactation.

Ihe analogue dị ọnụ ala site na 211 rubles.

Onye na-emeputa ihe: Oxford (India)
Mwepụta Mwepụta:

  • Mbadamba 20 mg, 30 PC.
Ntụziaka maka ojiji

Ọgwụ ọzọ dabere na kalịnda atorvastatin n'ụdị mbadamba. Ngwakọta nke Lipoford adịghị iche na Atoris, yabụ, ihe ndị na-egosi, contraindications na mmetụta ndị ọ na-enwe fọrọ nke nta ka ọ bụrụ otu.

Atomax (mbadamba) itute dochie Rating: 127 Top

Ihe analogue dị ọnụ ala site na 179 rubles.

Onye na-emepụta: Hetero Drags Limited (India)
Mwepụta Mwepụta:

  • Mbadamba 20 mg, 30 PC.
Ntụziaka maka ojiji

Atomax bu onye India dochie anya Atoris nwere otu nmehapu. Ọ na - emetụta ọgwụ ndị na - eme ka anwụ dị ala ma na - ejikwa otu DV. Contraindicated n'oge ime na lactation. Nsonaazụ ndị enwere ike, tupu ị gwa dọkịta nwere oge dị mkpa.

Analogs na ihe mejupụtara ma gosipụta maka ojiji

AhaỌnụahịa na RussiaỌnụahịa na Ukraine
Amvastan --56 UAH
Atorvacor --31 UAH
Vasocline --57 UAH
Livostor atorvastatin--26 UAH
Liprimar atorvastatin54 nkp57 UAH
Thorvacard 26 nkp45 UAH
Tulip Atorvastatin21 nkp119 UAH
Atorvastatin 12 nkp21 UAH
Limistin Atorvastatin--82 UAH
Lipodemin Atorvastatin--76 UAH
Litorva atorvastatin----
Pleostin atorvastatin----
Tolevas atorvastatin--106 UAH
Torvazin Atorvastatin----
Torzax atorvastatin--60 UAH
Etset atorvastatin--61 UAH
Aztor ----
Astin Atorvastatin89 nkp89 UAH
Atocor --43 UAH
Atorvasterol --55 UAH
Atotex --128 UAH
Novostat 222 nkp--
Atorvastatin-Teva Atorvastatin15 nkp24 UAH
Atorvastatin Alsi Atorvastatin----
Lipromak-LF atorvastatin----
Vazator atorvastatin23 nkp--
Atorem atorvastatin--61 UAH
Vasoclin-Darnitsa atorvastatin--56 UAH

N'elu ndepụta ọgwụ analogues, nke Atoris nọchiri, bụ nke kachasị mma n'ihi na ha nwere otu ihe mejupụtara nke ihe ndị na-arụ ọrụ ma na-emekọ ihe dabere na ngosipụta maka ojiji

Analogs site na ngosipụta na usoro eji

AhaỌnụahịa na RussiaỌnụahịa na Ukraine
Vabadin 10 mg simvastatin----
Vabadin 20 mg simvastatin----
Vabadin 40 mg simvastatin----
Vasilip simvastatin31 nkp32 UAH
Zokor simvastatin106 nkp4 UAH
Zokor Forte simvastatin206 rub15 UAH
Simvatin simvastatin--73 UAH
Vabadin --30 UAH
Simvastatin 7 nkp35 UAH
Vasostat-Health simvastatin--17 UAH
Vasta simvastatin----
Kardak simvastatin--77 UAH
Simvakor-Darnitsa simvastatin----
Simvastatin-zentiva simvastatin229 rub84 UAH
Simstat simvastatin----
Alleste --38 UAH
Zosta ----
Lovastatin lovastatin52 ikp33 UAH
Human rights pravastatin----
Leskol 2586 rub400 UAH
Leskol Forte 2673 nkp2144 UAH
Leskol XL fluvastatin--400 UAH
Crestor rosuvastatin29 nkp60 UAH
Mertenil rosuvastatin179 rub77 UAH
Klivas rosuvastatin--2 UAH
Rovix rosuvastatin--143 UAH
Rosart Rosuvastatin47 nkp29 UAH
Rosuvastatin Rosator--79 UAH
Rosuvastatin Krka rosuvastatin----
Rosuvastatin Sandoz Rosuvastatin--76 UAH
Rosuvastatin-Teva Rosuvastatin--30 UAH
Rosucard Rosuvastatin20 nkp54 UAH
Rosulip Rosuvastatin13 nkp42 UAH
Rosusta Rosuvastatin--137 UAH
Roxera rosuvastatin5 rub25 UAH
Romazik rosuvastatin--93 UAH
Romestine rosuvastatin--89 UAH
Rosucor rosuvastatin----
Rosuvastatin ngwa ngwa----
Calcium Acorta Rosuvastatin249 nkp480 UAH
Tevastor-Teva 383 nkp--
Rosistark rosuvastatin13 nkp--
Suvardio rosuvastatin19 nkp--
Redistatin Rosuvastatin--88 UAH
Rustor rosuvastatin----
Livazo pitavastatin173 rub34 UAH

Ngwakọta dị iche iche, nwere ike yikọ ọnụ na njiri na usoro nke ngwa

AhaỌnụahịa na RussiaỌnụahịa na Ukraine
Gemfibrozil Mpempe--780 UAH
Lipofen cf fenofibrate--129 UAH
Tricor 145 mg fenofibrate942 nkp--
Trilipix Fenofibrate----
Pms-cholestyramine nwere mmanụ oroma na-acha ọbara ọbara mgbe niile--674 UAH
Pumpkin Mkpụrụ Mmanụ Pumpkin109 nkp14 UAH
Ravisol Periwinkle obere, Hawthorn, Meadow clover, chestnutnut, White mistletoe, Sofora Japanese, Horsetail--29 UAH
Sicode mmanụ azụ----
Ngwakọta vitamin kadrum nke ọtụtụ ihe dị ike1137 rub74 UAH
Nchikota Omacor nke otutu ihe aru oru1320 nkp528 UAH
Azụ mmanụ azụ25 nkp4 UAH
Nchikota Epadol-Neo nke otutu ihe eji aru oru--125 UAH
Ezetrol ezetimibe1208 rub1250 UAH
Repata Evolokumab14 500 nkpUAH 26381
Praroent alirocoumab--28415 UAH

Etu esi achọta analog dị ọnụ ala nke ọgwụ na-akwụ ụgwọ?

Iji chọta analog na-enweghị ego ọfụma n’egwuregwu, mkpụrụ ọgụgụ ma ọ bụ ntụgharị, nke mbụ anyị na-atụ aro ị attentiona ntị na ihe mejupụtara ahụ, ya bụ otu ihe ahụ na njiri mara maka ojiji. Otu ihe eji eme ọgwụ eme ihe ga-egosi na ọgwụ ahụ kwekọrọ na ọgwụ ahụ, ọgwụ kwekọrọ ma ọ bụ ọgwụ ọzọ. Agbanyeghị, echefula maka ihe ndị na - adịghị ike nke ọgwụ ndị yiri ya, nke nwere ike imetụta nchekwa na ịdị irè. Echefula banyere ntuziaka nke ndị dọkịta, ọgwụ ịchọrọ onwe gị nwere ike imerụ ahụ ike gị, yabụ gbaa dọkịta gị mgbe niile tupu ị usingụ ọgwụ ọ bụla.

Omume ọgwụ

Atorvastatin bụ ihe nnọchianya nke ahụ sitere na otu nke statins. Mainzọ kachasị mkpa nke atorvastatin bụ mgbochi nke ọrụ HMG-CoA reductase, enzyme nke na-egbochi ntụgharị nke HMG-CoA na mevalonic acid. Mgbanwe a bụ otu n’ime ụzọ izizi na cholesterol (cholesterol) synthesis silsila n’ime ahụ. Mmechi nke Atorvastatin na cholesterol synthesis na - eduga n'ịbawanye ọrụ nke ndị na - anabata LDL na imeju, yana anụ ahụ extrahepatic. Ndị na-anabata ihe a na - ekekọta LDL ma wepụ ha na plasma ọbara, nke na - eduga n'ịbelata mkpokọta LDL-C n'ọbara.

Mmetụta antiatherosclerotic nke atorvastatin bụ nsonaazụ nke nsonaazụ ya na mgbidi nke arịa ọbara na akụkụ ọbara. Atorvastatin na-egbochi njikọ nke isoprenoids, nke bụ ihe na-eto eto nke mkpụrụ ndụ dị n’ime akwara ọbara. N'okpuru mmetụta nke atorvastatin, mmụba nke endothelium na-agbatị na akwara ọbara na-emeziwanye, ntinye nke cholesterol-LDL, apolipoprotein B, triglycerides (TG) na-ebelata, itinye uche nke cholesterol-HDL na apolipoprotein A.

Atorvastatin na-ebelata viscosity nke plasma ọbara na ọrụ nke ụfọdụ ihe coagulation na nchịkọta platelet. N'ihi nke a, ọ na - eme ka hemodynamics na - adịwanye mma ma na - edozi ọnọdụ nke coagulation system. Ndị na-egbochi HMG-CoA reductase na-emetụta metabolism nke macrophages, na-egbochi ọrụ ha ma na-egbochi nbibi nke oghere atherosclerotic.

Dịka iwu, nsonaazụ ọgwụgwọ nke atorvastatin na-etolite mgbe izu abụọ nke iji Atoris®, a na-enwetakwa mmetụta kachasị mgbe izu anọ gachara.

N'ụzọ dị oke mkpa belata ihe egwu nke nsogbu nsogbu ischemic (gụnyere ọnwụ site na infarction myocardial) site na 16%, ihe ize ndụ nke ịmaliteghachi ụlọ ọgwụ maka angina pectoris, yana ihe ịrịba ama nke ischemia myocardial, na 26%.

  • Mbelata nke cholesterol, cholesterol-LDL, apolipoprotein B na triglycerides n'ọbara ọbara nke ndị ọrịa nwere isi hyperlipidemia (ụdị Fredaịon IIa na IIb), gụnyere polygenic hypercholesterolemia, heterozygous hypercholesterolemia na hyperliplestidemia.
  • Mbelata nke nchịkọta cholesterol zuru oke, cholesterol-LDL na apolipoprotein B na ndị ọrịa nwere hyzycholesterolemia homozygous.
  • Atoris® na-eme ka itinye uche nke HDL-C n'ọbara ọbara ma belata ogo nke LDL-C / HDL-C.
  • A na-eji ya mee ihe maka enweghị ọgwụgwọ zuru ezu nke usoro ọgwụgwọ nri na ụzọ ọgwụgwọ ndị ọzọ na-abụghị ọgwụ ọgwụ.

Mgbochi Ọrịa Obi:

  • Ihe mgbochi mbu banyere nsogbu obi na ọrịa n’erughi ọrịa, ma enwere ọtụtụ ihe ọghọm maka mmepe ya: afọ kariri afọ 55, ihe nicotine riri ahụ, ọbara mgbali akwara, ọrịa shuga, ọkwa dị ala nke HDL-C na plasma ọbara, ịkọ mkpụrụ ndụ, gụnyere megide ndabere nke dyslipidemia.
  • Ihe mgbochi nke abụọ nke nsogbu obi na ọrịa obi na -arụ ọrịa iji belata ọnụ ọgụgụ ọnwụ, myocardial infarction, ọrịa strok, nwughari n'ụlọ ọgwụ maka angina pectoris na mkpa ịlọ ụwa.

Ihe ngbanwe

  • Ntinye obi na akụkụ nke ọgwụ ọ bụla.
  • Ọrịa imeju na-arụ ọrụ (gụnyere ịba ọcha n'anya na-adịghị ala ala, ịba ọcha n'anya ịba ọcha n'anya).
  • Imeju imeju.
  • Cirrhosis nke imeju nke etiology ọ bụla.
  • Mmụba na ọrụ nke usoro ịba ọcha n'anya nke mmalite amaghi site na ugboro atọ ma e jiri ya tụnyere VGN.
  • Ọkpụkpụ akwara Skeletal.
  • Enweghi ike nke Lactase, nnagide nke lactose, ọrịa glucose-galactose malabsorption syndrome.
  • Ime na oge inye nwa.
  • Afọ ruru afọ iri na asatọ (edobeghị ike na nchekwa iji ya).

Iji nlezianya: ahoụrụma, bụ akụkọ banyere ọrịa imeju.

Ime na lactation

Atoris® bụ mgbochi ime na n’oge a na-enye nwa ara. Nnyocha ụmụ anụmanụ na-egosi na ihe ize ndụ nke nwa ebu n’afọ nwere ike karịa uru ọ bụla ọ ga-abara nne.

N'ime ụmụ nwanyị toro nwa na-ejighị usoro ịtụkwasị obi nke igbochi afọ ime, a gaghị akwado iji Atoris® mee ihe. Mgbe ị na-eme atụmatụ ịtụrụ ime, ikwesiri ịkwụsị iji Atoris® opekata mpe ọnwa 1 tupu ịtụrụ ime gị.

Onweghi ihe akaebe banyere ikenye atorvastatin nwere mmiri ara. Agbanyeghị, n'ụfọdụ ụdị anụmanụ, nchịkọta nke atorvastatin n'ọbara na mmiri ara ara. Ọ bụrụ na ọ dị mkpa iji ọgwụ Atoris® n'oge ara, iji zere ihe ize ndụ nke ihe ojoo na ụmụ ọhụrụ, a ga-akwụsị inye ara ya.

Ntụziaka pụrụ iche

Tupu ịmalite Atoris®, a ga-enyerịrị onye ọrịa ahụ usoro hypocholesterolemic, nke ọ ga-agbaso n'oge usoro ọgwụgwọ niile.

Enwere ike ịhụbawanye na ọrụ nke enzymes hepatic n'ime ọbara ọbara n'oge ọgwụgwọ Atoris®. Mmụba a na-adịkarị obere ma ọ nweghị uru ọria. Agbanyeghị, ọ na-atụ aro ka nyochaa ọrụ nke enzymes imeju na ọbara n'ọbara tupu ọgwụgwọ, mgbe izu isii na nke iri na abụọ yana mmụba nke onorvastatin. Ọ bụrụ na mmụba okpukpu atọ na ọrụ nke ACT na / ma ọ bụ ALT dị ka HBV, a ga-akwụsị ịgwọ Atoris®.

Atorvastatin nwere ike ibute ọrụ CPK na aminotransferases.

N'ime ụmụ nwanyị toro nwa na-ejighị ọgwụ mgbochi a pụrụ ịdabere na ya, a gaghị akwado iji Atorisor eme ihe. Ọ bụrụ na onye ọrịa ahụ na-eme atụmatụ ịtụrụ ime, o kwesịrị ịkwụsị iwere Atoris® opekata mpe otu ọnwa tupu ịtụrụ ime amalite.

E kwesịrị ịdọ ndị ọrịa ọdụ na ha kwesịrị ịgakwuru dọkịta ozugbo ma ọ bụrụ na mgbu na-enweghị nkọwa ma ọ bụ adịghị ike nwere ahụ. Karịsịa ma ọ bụrụ na ha na-arịa ọrịa ịba ma ọ bụ ahụ ọkụ.

Withgwọ Atoris® nwere ike bute ọrịa myopathy, bụ nke rhabdomyolysis na - esochi, na - eduga n'ịda nnukwu akwara. Nsogbu nke nsogbu a na-abawanye mgbe ị na-ewere Atoris® otu ma ọ bụ karịa ọgwụ ndị a: ọgwụ fibroic acid, niacin, cyclosporine, nefazodone, ụfọdụ ọgwụ nje, antifungals azole, na nje HIV na-egbochi.

N'ime ngosipụta nke ọrịa myopathy, a na-atụ aro ka ekpebisi ike plasma nke CPK. Site na mmụba okpukpu iri na VHF nke ọrụ KFK, ọgwụgwọ Atoris® kwesịrị ịkwụsị.

Enwere akụkọ banyere mmepe nke atciic fasciitis na iji atorvastatin, agbanyeghị, njikọ na iji ọgwụ ahụ ga-ekwe omume, mana egosighi na etiology ahụ amabeghị.

E kwesịrị ịdọ ndị ọrịa ọdụ na ha kwesịrị ịgakwuru dọkịta ozugbo ma ọ bụrụ na mgbu na-enweghị nkọwa ma ọ bụ adịghị ike nwere ahụ, ọ bụrụ na ọnya ma ọ bụ ahụ ọkụ na-eso ya.

Atoris® nwere lactose, yabụ ojiji nke ndị ọrịa nwere ụkọ lactase, nnagide nri nke lactose na ọrịa glucose-galactose malabsorption.

Mmetụta ikike ịkwọ ụgbọ ala ma jiri usoro rụọ ọrụ.

Nyere ohere i nwere ino ilu, a gha akpachara anya mgbe inya ugboala na ngwa oru ndi ozo choro itinye uche nlebara anya na osiso nke mmeghachi omume psychomotor.

Mbadamba otu 1 nwere:

Arụ Ọrụ: atorvastatin calcium 10.36 mg, (ihe ruru 10 mg atorvastatin, otu isi).

Ndị e mere: povidone - 5.8 mg, sodium lauryl sulfate - 2.9 mg, calcium carbonate - 31.84 mg, MCC - 29 mg, lactose monohydrate - 57.125 mg, ssumum croscarmellose - 7.25 mg, magnesium stearate - 0.725 mg.

N'ọbọ ihe nkiri: Opadry II HP 85F28751 ọcha (mmanya polyvinyl, titanium dioxide (E171), macrogol 3000, talc) - 4.35 mg.

Usoro onunu ogwu na nhazi

N'ime, n'agbanyeghị nri.

Tupu ịmalite ị Atụ ọgwụ Atoris®, a ga-ebugharị onye ọrịa ahụ na nri nke na -ebelata mbelata nke egbugbere ọnụ ọbara, nke a ga-ahụrịrị n'oge ọgwụgwọ ya dum. Tupu ịmalite usoro ọgwụgwọ, ị kwesịrị ịgbalị iji nweta nchịkwa nke hypercholesterolemia site na mmega ahụ na oke ibu na ndị ọrịa nwere oke ibu, yana ọgwụgwọ maka ọrịa na-akpata.

Ọgwụgwọ ebido na usoro akwadoro ọgwụ nke 10 mg. Ọgwụ nke ọgwụ ahụ dị site na 10 ruo 80 mg otu ugboro kwa ụbọchị ma ahọpụtara na-eburu n'uche ntinye uche mbụ nke LDL-C, ebumnuche nke ọgwụgwọ na mmetụta ọgwụgwọ nke onwe ya.

Enwere ike iwere Atoris once otu oge n'oge ọ bụla n'ụbọchị, mana n'otu oge kwa ụbọchị. A na-achọpụta mmetụta ọgwụgwọ ahụ ka izu abụọ nke ọgwụgwọ gasịrị, na nsonaazụ kachasị na-etolite mgbe izu anọ gachara. Ya mere, usoro onunu ogwu ekwesighi igbanwe tupu izu anọ abidola ọgwụ bidoro n ’ọgwụ ị na -ebu.

Na nmalite ọgwụgwọ na / ma ọ bụ n'oge mmụba nke dose, ọ dị mkpa iji nyochaa ịta nke lipids na plasma ọbara kwa izu 2-4 ma mezie ọnụọgụ ya.

Ihe mbu (heterozygous hereditary na polygenic) hypercholesterolemia (ụdị IIa) na hyperlipidemia agwakọta (ụdị IIb): ọgwụgwọ na-amalite site na usoro ọgwụgwọ akwadoro, nke a na-abawanye ka izu anọ gachara, dabere na nzaghachi onye ọrịa. Oke kachasị kwa ụbọchị bụ 80 mg.

Homozygous hereditary hypercholesterolemia: ụdị ọgwụgwọ ahụ bụ otu ihe ahụ na ụdị hyperlipidemia ndị ọzọ. A na-ahọrọ usoro izizi otu n’otu, dabere ogo ọrịa ahụ. N'ime ọtụtụ ndị ọrịa nwere hypercholesterolemia homozygous, a na-ahụ mmetụta kachasị mma site na iji ọgwụ ahụ na ọgwụ kwa ụbọchị nke 80 mg (otu oge). A na-eji Atoris® agwọ ọrịa na usoro ọgwụgwọ ndị ọzọ (plasmapheresis) ma ọ bụ dịka ọgwụgwọ bụ isi ọ bụrụ na ọgwụgwọ na ụzọ ndị ọzọ agaghị ekwe omume.

Otu ndị ọrịa pụrụ iche.

Ndị okenye na-arịa ọrịa.

N'ime ndị ọrịa meworo agadi, a gaghị agbanwe ọgwụ Atoris®.

Alrụ ọrụ na-arụ ọrụ na ụlọ.

Ọ naghị emetụta mkpokọta nke atorvastatin na plasma ọbara ma ọ bụ ogo nke mbelata nke mkpokọta LDL-C site na iji atorvastatin, ya mere, a chọghị ịgbanwe ọgwụ a chọrọ.

Ọrụ imeju na-arụ ọrụ.

N'ime ndị ọrịa nwere ọrụ imeju na-arụ ọrụ, ọ dị mkpa ịkpachara anya (n'ihi nkwụsị nke ọgwụ iji wepụ ahụ). N'ọnọdụ dị otú a, a ga-eji nlezianya nyochaa ụlọ ọgwụ na nyocha ụlọ nyocha (ị na-ahụ maka ọrụ ACT na ALT) mgbe niile. Site na mmụba dị ukwuu na transpeases hepatic, a ga-ebelata ọgwụ Atoris® ma ọ bụ kwụsị ọgwụgwọ.

Jiri na ọgwụ ndị ọzọ.

Ọ bụrụ na ọ dị mkpa, na ojiji nke cyclosporine kwa ụbọchị nke ọgwụ Atoris® ekwesịghị gafere 10 mg.

Atoris - ozi izugbe

Onye na-ahụ maka hypolipPs Atoris (Atoris) bụ akụkụ nke otu nke akpụ akpụ na-egbochi ịrụ ọrụ nke enzyme n'ime imeju (HGM-CoA), bụ ọrụ maka mmepụta cholesterol.

A na-emepụta ọgwụ ahụ n'ụdị mbadamba n'ụdị dị iche iche: 10 mg, 20 mg na 40 mg nke ihe mejupụtara atorvastatin. Otu mbadamba ihe nwere obere nke excipients - povidone, sodium lauryl sulfate, magnesium stearate, lactose monohydrate, wdg.

Usoro nke ị ofụ ọgwụ ahụ jikọtara ya na njikọta cholesterol njikọta yana ịba ụba nke ndị na-anabata LDL na anụ ahụ extrahepatic na imeju. Na-esote, ndị na-anabata ihe na-ekekọta LDL irighiri ihe, na-ewepụ ha n'ọbara. N'ihi ya, a na-ebelata cholesterol ọbara.

Dọkịta nyere Atoris iwu n ’ụdị okwu ahụ:

  • ndị ọrịa na-enweghị ọrịa akwara obi ha n'ụlọ ọgwụ iji belata ihe egwu infarction myocardial, ọrịa strok, angina pectoris na mkpa maka usoro mwekọ ịkpụgharị myocardial,
  • ndị ọrịa na-arịa ọrịa shuga na-abụghị insulin na-arịa ọrịa shuga mellitus (ụdị 2) na-enweghị ọrịa obi na-egosipụta ọrịa obi iji belata ohere nke nkụchi obi na ọrịa strok,
  • ndị ọrịa nwere ọrịa obi na -akpọpụta akwara iji wee belata ọghọm ọrịa myocardial na-abụghị nke na-egbu egbu, ọrịa na-egbu egbu na-adịghị egbu egbu, angina pectoris, mkpa maka ịmụgharị myocardial na ụlọ ọgwụ n'ihi nkụchi obi.
  • dị ka mgbakwunye na nri pụrụ iche maka isi (ezinụlọ / ndị na-abụghị ezinụlọ) na agwakọta (ụdị IIa na IIb) hypercholesterolemia,
  • dị ka mgbakwunye nri maka hypertriglyceridemia (ụdị IV), isi dysbetalipoproteinemia (ụdị III), yana homozygous familial hypercholesterolemia,
  • ndị ọrịa dị afọ iri na asatọ ruo iri na abụọ nwere akụkọ gbasara ezinụlọ nke akwara gbasara ọrịa mbụ ma ọ bụ karịa ihe abụọ maka mmepe ha.

Atoris nwere ọnụ ọgụgụ dị nta nke contraindications. N'etiti ha, ọ dị mkpa iji gosipụta adịghị mma na njikọ nke mbadamba, afọ ime na lactation, nsị nke imeju na ọkwa dị elu nke transaminases.

Nnukwu analogues na nnọchi ọgwụ ọjọọ atoris maka ụmụaka na ndị okenye

Atoris bu ogwu nke mbubata si. Analogues dị ọnụ ala karịa Atoris nwere otu ma ọ bụ ihe yiri ya na-arụ ọrụ, a na-emepụta ya na mba dị iche iche, gụnyere ndị na-emepụta ụlọ. Ọgwụ n'onwe ya na Russia na-akwụ ihe ruru 400 - 1000 rubles. Mgbanwe a dị na ọnụahịa bụ n'ihi ọdịiche nke mbadamba ụrọ dị na ngwugwu yana usoro ha nke ihe arụ ọrụ.

Ngosipụta nke iji gosipụtara ihe na-ekwekọghị nye ndị na-azụ ahịa okwu ahụ hyperlipidemia. N'ezie, nke a pụtara mmụba nke ọkwa lipids n'ime ọbara (dịka ọmụmaatụ, enwere ike ịkpọ cholesterol, mana enwere ọtụtụ ihe), ihe ndị a bụ ihe dị iche iche na-enweghị mkpụrụ ndụ na - enweghị ike ịbanye n'ime ọbara ma nwee ike imechi ọnya vaskụla.

Ọnụnọ ha gosipụtara mmebi nke metabolism abụba. Ọgwụ dị iche iche nwere ike wepu lipids n'ọbara ma belata ọkwa ha.

Increasedba ụba nke itinye n'ọrụ bụ ihe kwesịrị ekwesị maka ndị ọrịa nwere ọrịa dị oke njọ.

Analogs nke mmepụta Russian

Mkpụrụ ọgwụ analogues dị ọnụ ala nke ndị na-emepụta ụlọ na-enwe ike ịnagide mmụba nke ọkwa nke lipid. Ma ọ bụghị mgbe niile ọgwụ dị ọnụ ala karịa dị iche na njirimara mma. Na tebụl dị n'okpuru ebe a, anyị depụtara ihe ndị kachasị ọsọ.

Aha ọgwụỌnụ ego dị na rublesNjirimara
Cardiostatin251-300Erere maka ọgwụgwọ nke ọrịa obi na - ebute oke cholesterol n'ime ọbara. A na-akọwa ntụzi aka nke ojiji eji ntuziaka ahụ.
Rosuvastatin500-1000Edere ya naanị ka ọ bụrụ nkwụba ọzọ maka nri hypercholesterolemia ma ọ bụ hypertriglyceridemia.
Simvastatin200-600Ọ bụ ndị nrụpụta Russia na-emepụta ya ozugbo, otu onye na-emepụta dị na Czech Republic. Ọgwụ nwere nnukwu ndepụta nke contraindications. Amachibidoro ya n’oge ime.
Atomax385-420Onwere onye India na -eme otu aha. Lowers cholesterol, mana naanị na njikọta na nri dị mma na ịnabata mmachibido iwu nri ndị nwere abụba.
Atorvastatin150-180Mmekọrịta dị ọnụ ala maka mmepụta Russian. Ruo ihe dị ka afọ 18 ka a na-atụghị ọgwụ ọ bụla, ị ofụ ọgwụ ga-ekwe omume naanị ma ọ bụrụ na esoro ihe oriri.
Novostat302-350Onu ogugu egosi ihe eji eme ya, na enye ya bu mmanye. Tupu ịmalite oriri ahụ, a na-atụ aro idobe nri siri ike.

Ndị nnọchi Ukraine

Ndepụta nke analogues nke Yukiren mejupụtara nwere nkwadebe eke. Dochie ọgwụ dị ọnụ ala bụ ihe amamihe dị na mbido ọrịa ahụ ma ọ bụ dịka ngwa ọzọ.

  1. Cholesterol Alfalfa. Ọgwụ a, nke emere na ntọala sitere na ebumpụta ụwa, dị mma maka ndị na-eto eto na ndị okenye. Nabatara site na ọmụmụ. Ọ na-efu 210 rubles.
  2. Aterovit. Na-enyere aka mee ka arịa ọbara na cholesterol dị ala. Ngwakọta ọgwụ a bụ ihe okike. Ha ruru 140 rubles.
  3. Cardiochistin. Edere ya maka cholesterol dị elu. Meziwanye ahụike na atherosclerosis. Amachibidoro ị drugụ ọgwụ a n’oge ime na n’oge a na-enye nwa ara. Ọ na-efu 200 rubles.
  4. Mgbakwunye Omega Plus. Ome zuru oke nke Omega acid nke ụdị 3 na 6. Na-ahụ maka ọrụ sistem nke obi. Anabataghị ịmalite nke ọgbụgba ọbara. A nwalere ọgwụ a n'ụlọ ọgwụ. Ọnụahịa ahụ na Russia bụ 330 rubles.
  5. Dioscorea Plus. Lowers cholesterol na-ebelata ọbara mgbali elu. Na-echebe arịa ọbara site na mmebi. Ngwakọta zuru oke. Ọ na-efu ihe dịka 250 rubles.

Ọkpụkpụ Belarusia

Ọkpụkpụ Belarus adịghị ọnụ. Ndị a bụ ndị nọchiri anya ihe dị iche iche na-arụ ọrụ na usoro dị iche iche nke ekpughere ahụ onye ọrịa.

Aha ọgwụỌnụ ego dị na rublesNjirimara
Lovastatin130-150A na-emepụta ọgwụ ahụ na Ukraine na Masedonia. Ọ na-agwọ ụdị hypercholesterolemia nke 2 na nke 3 ka edepụtara ya maka ndị ọrịa nwere atherosclerosis. Tupu ojiji, ọ na-atụ aro iji nlezianya mụọ ndepụta ọgwụ ọgwụ na-emekọrịta ihe na-emetụta ahụike nke onye ọrịa.
Aterol714-750Ọ na - ewepu nsị na toxins, belata cholesterol. Adabara mgbochi nke atherosclerosis. Ihe mebere eke.
Choledol700-750Nkwụsị mmachi maka nchịkwa ọnụ. Dọ aka na ntị megide nkụchi obi, ọrịa strok. Normalizes lipid metabolism. Ngwakọta ahụ gụnyere ihe ndị sitere n'okike.
Osisi ogwu ogwu nke China1700-1800Agbakwunye nri. Ọ na-ebelata agụụ, na-ewepụ oke mmiri, toxins na toxins n'ahụ. Na-akwalite ibu felata. A na-etolite ihe mejupụtara ahụ site n'ụkpụrụ ndị China na usoro ahụike n'ihi ihe ọkụkụ sitere n'okike. Teknụzụ ọgbara ọhụrụ wetara ha izu-ike.

Lomụ amaala mba ọzọ

Ọgwụ ndị e webatara dị ọnụ. Nhọrọ kachasị mma edepụtara maka ikpe ọ bụla bụ nke onwe ya. Emere mkpebi kacha mma yana dọkịta. Asọfọ Atoris nwere njirimara nke ha.

  • Vasilip. A na-eme ya na Slovenia. Adabara ndị ọrịa shuga. Normalizes cholesterol, mana ọ bụ naanị na nri. Dabere na ọnụọgụ mbadamba ihe dị na ngwugwu ahụ, ọ na-efu site na 160 ruo 340 rubles.
  • Zokor. Emere ya na Netherlands. Theụ ọgwụ ahụ wee bụrụ ihe dabara adaba mgbe enwere nnukwu ihe ize ndụ nke ịmalite ọrịa obi. Erere na-eri 750 rubles.
  • Crestor. Emere na UK. Kwesịrị ekwesị maka ndị ọrịa nwere atherosclerosis ma ọ bụ ụdị hypercholesterolemia dị iche iche.Ọnụahịa ọgwụ nke ọgwụ dịgasị iche iche sitere na 700 ruo 3600 rubles.
  • Rosulip. Emere na Hungary. Anaghị anabata nguzobe cholesterol. A na-ahapụ ya naanị site na ndenye ọgwụ. Ofzọ iche nke mbadamba nkume si na 700 ruo 1200 rubles.
  • Mertenyl. A na-eme ya na Hariari. Mmetụta na ụmụaka nwere ọgwụ a amụbeghị amụ ma ọ machibidoro ịkọ ya ụmụaka. A na-ere ọgwụ dị iche iche, ọnụahịa ha na-amalite site na 700 rubles wee rute 1400 rubles.
  • Rosucard. Czech Republic Ihe mejupụtara ọgwụ ahụ gụnyere rosuvastatin na-arụ ọrụ. Ntinye akwụkwọ ga-ekwe omume naanị mgbe emechara dọkịta. Otu ọgwụ dị ọnụ ala dị ọnụ ala, ọnụahịa ya anaghị aga 500 rubles.

Otu esi edochi atoris dị mfe idozi. Enwere otutu analogues. Ọnụahịa ha dị iche iche, ndepụta ihe na-egosi dị iche iche, enwere ọgwụ ọgwụ nwere nnukwu mmetụta na anụ ahụ, enwere ndị a na-eduzi.

A na-ahuta ogwu di nma karie mgbe omumu omumu zuru oke na laabula ma obu ulo ogwu.

Mbadamba Atoris: ntuziaka maka ojiji, mmetụta ndị ọzọ, analogues, ọnụahịa, nyocha

Atoris ọgwụ, ntuziaka maka enyere nke a na-enye ndị na-agụ akwụkwọ anyị, bụ nke ọgwụ ọgwụ belata, nke bụ ọgbọ nke atọ - ọgwụ na - enyere aka belata mkpụkọ nke obere lipoproteins (LDL) - nke a na - akpọ 'cholesterol ọjọọ' - na membranes cell, anụ ahụ na gburugburu ebe obibi. ọbara, akwara ozi, mmiri mkpụrụ ndụ, ọria ọbara (akụkụ ahụ na mmiri).

Ojiji nke ụdị a na-ebelata ohere nke ọrịa obi na ndị ọrịa nọ n'ọgbọ dị n'etiti, ọ bụ ezie na ndị mmadụ karịrị afọ iri asaa anaghị ekwupụta usoro a.

A na-atụ aro ka eji rụọ ọrụ ahụ naanị n'ọnọdụ ụfọdụ ebe usoro mgbochi mgbochi (na-agbaso nri cholesterol dị ala, egwuregwu oge niile na ihe omume iji belata ahụ mmadụ) enyeghị aka na normalization nke lipid metabolism.

Ihe omuma banyere ihe mejuputara, udiri mpempe na ngwugwu

Atoris nwere otu usoro onunu ogwu ma dị n'ụdị ọcha - ntakịrị biconvex - mbadamba okirikiri nwere mkpuchi ihe nkiri. Ihe na - arụ ọrụ nke ọgwụ a bụ atorvastatin.

Ọdịnaya dị n’ime mbadamba ụrọ nke ọ bụla nwere ike ịbụ: 10, 20, 30, 40, 60 na 80 mg.

A na-ewepụta ihe ndị ọzọ nke mejupụtara kemịkal:

  • Microcrystalline cellulose,
  • Sodium sulfur sulfate,
  • Steeti magnesium,
  • Kaadị carbon
  • Lactose conohydrate,
  • Povidone
  • Crospovidone
  • Croscarmellose sodium.

Emeputara n'ọbọ ihe nkiri Opadry II:

  • Tal,
  • Titanium dioxide (ihe mgbakwunye nri E171),
  • Polyethylene glycol (n'ụzọ ụfọdụ a na-akpọ ya macrogol-3000 ma ọ bụ mgbakwunye nri E1521),
  • Polyvinyl mmanya.

Ihe dị mkpa nke mbadamba ihe dị na mmebi ahụ yiri ihe dị ọcha na-acha ọcha nke nwere akụkụ siri ike. Mpempe ngwongwo dị (blisters) na mbadamba nkume na-etinye n'ime ngwugwu kaadiboodu.

Dabere na nchikota nke oke arụ ọrụ, ngwugwu nke ọ bụla nwere ike ịnwe mbadamba iri ruo iri itoolu. Ntuziaka maka iji ya ga-ejikọrịrị na ngwugwu ọ bụla na ọgwụ.

Njirimara nke pharmacodynamics

Ngwurugwu atoris, nke nke otu statins, nwere mmetụta dị ala na-egbu egbu n'ihi ikike nke ihe arụ ọrụ na-arụ ọrụ, atorvastatin, igbochi (jiri nwayọ) ọrụ nke enzyme pụrụ iche (HMG-CoA reductase), nke na-ekere òkè na mbido mbụ nke cholesterol synthesis nke mkpụrụ ndụ imeju na-eme (hepatocytes) )

Site na ntinye nke atorvastatin, a na-ebelata oke cholesterol nke hepatocytes, na-enye ntinye aka na mbido mmụba ọnụ ọgụgụ nke ndị na-anabata LDL site na njide na ojiji nke obere lipoprotein cholesterol dị ugbu a n'ọbara.

N'okwu a, metabolism nke lipoproteins, nke gụnyere apolipoprotein - protein apoB, nke bu cholesterol “ọjọọ” na nke ndị LDL nabatara nke mkpụrụ ndụ imeju na-abawanye.

N'ihi usoro ndị dị n'elu, iberibe lipoproteins dị mkpụmkpụ, nwere obere oge, ewepụrụ ya oge ụfọdụ na plasma ọbara, nke pụtara na ọ na-agbadata ọkwa nke obere lipoprotein cholesterol dị ala.

N'ihi nke a pụrụ isi kwuo:

  • Mgbupu umu ihe ndi ozo di iche-iche - isoprenoids guzobere n’ahu mmadu site na acetic
  • Acids na sel na-akwalite sel na-akpụ akpụ akpụ intravaskụla,
  • Ngkwado ntụrụndụ nke ndabere endothelium,
  • Ibelata triglycerides, protein apoB na obere protein lipoprotein cholesterol,
  • Mmụba na mkpokọta apolipoprotein AI (protein apoA-I) na lipoproteins dị elu, nke bụ ihe na-ebu “ezigbo cholesterol”,
  • Ọbara plasma ọbara dara mgbada
  • Nwepu nke usoro nke coagulation na gluing (nchịkọta) nke platelet,
  • Imeziwanye hemodynamics (mmegharị ọbara site na sistemụ akwara ọbara site na mpaghara mgbali elu na mpaghara ala),
  • Normalization nke ọbara coagulation usoro,
  • Ing igbochi oke arụ ọrụ nke macrophages (mkpụrụ ndụ maka ijide na nhazi nke nje bacteria, mkpụrụ ndụ nwụrụ anwụ yana akụkụ ahụ), nke na - enyere aka igbochi mbibi nke usoro akpọrọ atherosclerotic plaques.

A na-achọpụta nsonaazụ mbụ nke ekpughere atorvastatin mgbe izu abụọ nke ị theụ ọgwụ ahụ gasịrị, na-eru ụkpụrụ kachasị mgbe otu ọnwa gasịrị. N'ime usoro ịgwọ ọrịa, emere ka ọ pụta ìhè na atoris bụ ọgwụ ị nwere ike ịbelata belata ọrịa ischemic, mkpa ọ dị ịnwe ụlọ ọgwụ na ọnụọgụ ndị nwụrụ.

Mlọ ọgwụ

  • Observed na-ahụkarị ọgwụ ọjọọ atoris na plasma ọbara n'ime awa 1-2 ka ewerechara mbadamba ihe ndị ahụ.
  • Aclọ ọgwụ ọgwụ nke atorvastatin abụghị nke nwoke ma ọ bụ afọ ole ndị ọrịa dị.
  • Achoputara na aru ndi oria na egbu egbu nke imeju, onu ogugu nke atorvastatin di elu karie iri na isii.
  • Mgbe e risịrị nri, ọnụego mmịpụta (nnabata) nke ọgwụ na-ebelata ntakịrị, n’agbanyeghi ọkwa nke lipoprotein cholesterol dị obere anaghị agbanwe ma ọlị.
  • Nnukwu bioavailability nke atorvastatin, nke bu ụzọ gafere na imeju onye ọrịa, dị ala: ọ bụ ihe karịrị 12% (a kọwara ya site na ịdị ukwuu nke usoro metabolic). Usoro bioavailability nke mmetụta mgbochi nke atorvastatin na HMG-CoA reductase dị nso na 30%.
  • Mmekọrịta nke ihe mejupụtara ọgwụ ọgwụ a na protein protein plasma bụ 98%.
  • Atorvastatin anaghị emeri ihe mgbochi nke ụbụrụ ọbara, metabolism ya na-abụkarị n'ụdị imeju n'ihi ikpughe cytochrome P4503A4. Metabolites na-arụ ọrụ metabolites guzobere n'ihi usoro a na-enye akụkụ buru ibu (ihe dị ka 70%) nke ọgwụ ọgwụ Atoris, nke na-ewe awa iri abụọ na atọ.
  • Ọkara ọkara nke ọgwụ ahụ bụ ihe dị ka awa iri na anọ. Imirikiti ọgwụ na-ahapụ ahụ onye ọrịa ahụ bile, ntakịrị dị ntakịrị (ihe dịka 45%) - na ọnya. Site na mmamịrị, ọ bụghị ihe karịrị 2% ọgwụ a kapịrị.

Atoris - analogues

Iji belata ọkwa nke triglycerides, lipids na cholesterol na plasma ọbara, a na-atụpụta statins. Atoris na-ekwu maka ha - achọrọ analogues nke iji ọgwụ ahụ eme ihe ma ọ bụrụ na anabataghị ọgwụ a ma ọ bụ, n'ihi ihe ụfọdụ, ọ gaghị ekwe omume ịzụta ya. Ọ dị mma ịmara na ọtụtụ mkpụrụ ndụ ihe omimi dị ọnụ ala karịa.

Analogues nke ọgwụ Atoris

Emeputara nhazi a gosipụtara na ndabere nke calcium atorvastatin - ihe emebere iji belata ntinye nke lipids n'ime ọbara. Atoris na-arụpụtakwa ọgwụ antisclerotic na mgbidi nke arịa ọbara, na-ebelata viscosity na njupụta nke plasma, na-eme ka hemodynamics dịkwuo mma, na-ebelata ohere nke ibute ọrịa obi.

Ọgwụ ndị a nwere mmetụta na ihe mejupụtara:

  • Torvalip
  • Ihe eji agwu Tulip
  • Torvas
  • Liptonorm,
  • Thorvacard
  • TG-tor
  • Torvazin
  • Atorvastatin
  • Liprimar
  • Atorvox
  • Lipoford
  • Vazator
  • Lipona
  • Amvastan
  • Astin
  • Atocor
  • Atorvacor
  • Atotex
  • Atorvasterol,
  • Atormak
  • Lipodemin,
  • Limistin
  • Lipimax
  • Vasocline
  • Livostor
  • Torvazin
  • Lithuania,
  • Tolevas
  • Etset,
  • Torzaks,
  • Actastatin
  • Abisiak
  • Aztor
  • Liperosis
  • Storvas
  • Escolan
  • Emstat
  • Torvadak
  • Lipitin,
  • Atrok.

Kedu nke kachasị arụ ọrụ ma rụọ ọrụ ka mma - Atoris ma ọ bụ Torvakard?

Mkpụrụ ọgwụ abụọ a na-atụle na-esite n'otu ahụ arụ ọrụ, ihe mejupụtara ihe ndị ọzọ eji arụ ọrụ bụkwa otu. Cardiologists kwenyere na enweghi ọdịiche dị egwu n'etiti ọgwụ ndị ahụ, naanị ihe dị iche na ọnụahịa bụ na Torvard dị ntakịrị ọnụ ala, ọbụlagodi na ntinye uche kachasị (40 mg).

Kedu nke ka mma ịzụta - Atorvastatin ma ọ bụ Atoris?

Ọgwụ ndị a nwekwara otu ihe mejupụtara, ụdị ntọhapụ yana ọdịnaya nke ihe ndị mejupụtara ya. A na-ahọrọ Atorvastatin karịa, ebe ọ bụ na ọ ka anabata karịa ma na-akpata mmetụta ndị dị ntakịrị. N'okwu a, ihe nnọchianya ahụ dị ọnụ ahịa karịa Atoris, nke ọkwa dị elu kọwapụtara na ntinye nke mbadamba ihe.

Krestor ma ọ bụ Atoris - nke ka mma?

Ọgwụ mbụ egosipụtara sitere n’ihe ọzọ - rosuvastatin. Ọ na - arụ ọrụ yiri Atoris, mana ọ na - a belata obere usoro, ebe 5 mg nke rosuvastatin kwekọrọ na ike nke 10 mg nke atorvastatin.

Ya mere, a na-ahụta Krestor ka ọ bụrụ ọgwụ dabara adaba, nke enwere ike ịkarị obere oge. N'otu oge, ọ na-efu karịa Atoris, ihe dị ka ugboro 2,5.

Atoris ma ọ bụ Liprimar dị irè karị, oleekwa ihe dị mma ịzụta?

A na-eme ọgwụ ndị atụnyere na ndabere nke atorvastatin. N'ime uru nke Liprimar bara uru ịmara:

  • ọnụọgụ ọgwụ ndị dịnụ (10, 20, 40 na 80 mg),
  • nhicha nke kachasi nma, nke n’enwe obere ihe ojoo.
  • ezigbo ndidi
  • elu bioavailability na digestibility.

Ka o sina dị, Liprimar adịkarịghị edepụtara ya n'ihi ọnụahịa dị oke elu, ọ dị 4.5 ugboro karịa Atoris.

Kedu ihe dị mma ị toụ mmanya - Atoris ma ọ bụ Simvastatin?

Ọgwụ ndị ahụ a tụrụ aro nwere ihe dị iche iche na-arụ ọrụ, yana iji nweta mmetụta ọgwụgwọ achọrọ nke simvastatin, achọrọ 20 mg, ebe atorvastatin chọrọ 10 mg.

Onweghị ọdịiche dị n'etiti ọgwụ, belụsọ maka ụdị ọnụahịa ha. Atoris ji ihe dị ka okpukpu 4 karịa ọnụ. Mgbe ị na-ahọrọ n'etiti ya na Simvastatin, ọ dị mkpa iburu n'uche njirimara onye ọrịa ahụ, ọnụnọ nke mmeghachi ahụ nfụkasị na mmụba na akụkụ nke ọgwụ.

Roxer ma ọ bụ Atoris - nke ka mma?

Nhazi nke ọgwụ ndị a dịkwa iche, roxuvastatin bụ ntọala nke Roxers. Dịka anyị kwurula, ọkacha mma maka ihe a, ebe ọ bụ na ọ ka arụ ọrụ karịa, anaghị achọ nchịkwa ugboro ugboro yana nnukwu ọgwụ. Ọtụtụ ndị dọkịta depụtara Roxer ọtụtụ oge, n'ihi na ọgwụ a, na mgbakwunye na arụmọrụ, dị ọnụ ala, ọ dị ọnụ ala karịa 2 Atoris.

Atoris analogues na onu ahia

Tupu ịmalite Atoris®, a ga-enyerịrị onye ọrịa ahụ usoro hypocholesterolemic, nke ọ ga-agbaso n'oge usoro ọgwụgwọ niile.

Enwere ike ịhụbawanye na ọrụ nke enzymes hepatic n'ime ọbara ọbara n'oge ọgwụgwọ Atoris®. Mmụba a na-adịkarị obere ma ọ nweghị uru ọria.

Agbanyeghị, ọ na-atụ aro ka nyochaa ọrụ nke enzymes imeju na ọbara n'ọbara tupu ọgwụgwọ, mgbe izu isii na nke iri na abụọ yana mmụba nke onorvastatin.

Ọ bụrụ na mmụba okpukpu atọ na ọrụ nke ACT na / ma ọ bụ ALT dị ka HBV, a ga-akwụsị ịgwọ Atoris®.

Atorvastatin nwere ike ibute ọrụ CPK na aminotransferases.

N'ime ụmụ nwanyị toro nwa na-ejighị ọgwụ mgbochi a pụrụ ịdabere na ya, a gaghị akwado iji Atorisor eme ihe. Ọ bụrụ na onye ọrịa ahụ na-eme atụmatụ ịtụrụ ime, o kwesịrị ịkwụsị iwere Atoris® opekata mpe otu ọnwa tupu ịtụrụ ime amalite.

E kwesịrị ịdọ ndị ọrịa ọdụ na ha kwesịrị ịgakwuru dọkịta ozugbo ma ọ bụrụ na mgbu na-enweghị nkọwa ma ọ bụ adịghị ike nwere ahụ. Karịsịa ma ọ bụrụ na ha na-arịa ọrịa ịba ma ọ bụ ahụ ọkụ.

Withgwọ Atoris® nwere ike bute ọrịa myopathy, bụ nke rhabdomyolysis na - esochi, na - eduga n'ịda nnukwu akwara.

Nsogbu nke nsogbu a na-abawanye mgbe ị na-ewere Atoris® otu ma ọ bụ karịa ọgwụ ndị a: ọgwụ fibroic acid, niacin, cyclosporine, nefazodone, ụfọdụ ọgwụ nje, antifungals azole, na nje HIV na-egbochi.

N'ime ngosipụta nke ọrịa myopathy, a na-atụ aro ka ekpebisi ike plasma nke CPK. Site na mmụba okpukpu iri na VHF nke ọrụ KFK, ọgwụgwọ Atoris® kwesịrị ịkwụsị.

Enwere akụkọ banyere mmepe nke atciic fasciitis na iji atorvastatin, agbanyeghị, njikọ na iji ọgwụ ahụ ga-ekwe omume, mana egosighi na etiology ahụ amabeghị.

E kwesịrị ịdọ ndị ọrịa ọdụ na ha kwesịrị ịgakwuru dọkịta ozugbo ma ọ bụrụ na mgbu na-enweghị nkọwa ma ọ bụ adịghị ike nwere ahụ, ọ bụrụ na ọnya ma ọ bụ ahụ ọkụ na-eso ya.

Atoris® nwere lactose, yabụ ojiji nke ndị ọrịa nwere ụkọ lactase, nnagide nri nke lactose na ọrịa glucose-galactose malabsorption.

Mmetụta ikike ịkwọ ụgbọ ala ma jiri usoro rụọ ọrụ.

Nyere ohere i nwere ino ilu, a gha akpachara anya mgbe inya ugboala na ngwa oru ndi ozo choro itinye uche nlebara anya na osiso nke mmeghachi omume psychomotor.

Atoris: ntuziaka maka ojiji, analogues na nyocha

Atorvastatin belata plasma cholesterol na mkpokọta lipoprotein site na igbochi GMK-CoA reductase, na-esote site na biosynthesis nke cholesterol n'ime imeju, na-emekwa ka ọnụ ọgụgụ nke ndị na-anabata heDatic LDL na cell, nke na-eduga n'ịba ụba uptake na LDL catabolism.

Na-ebelata nguzobe LDL na onu ogugu nke LDL. Atoris na-ebute mmụba na-adịgide adịgide na ọrụ nke ndị na-anabata LDL na mgbakwunye mgbanwe dị mma na ogo nke LDL ahụ na-ekesa.

Nke ọma na-ebelata LDL cholesterol na ndị ọrịa nwere hypercholesterolemia homozygous familial, na nke a bụ otu na-azabeghị ọgwụ ịba ụba mmadụ.

N'okwu dị mfe, ojiji nke Atoris na-enyere aka ịkwụsị mmepụta cholesterol n'ime ahụ, belata ọnụ ọgụgụ dị ala nke lipoprotein cholesterol na imeju.

Mmetụta ọgwụgwọ na-etolite izu 2 mgbe mmalite nke ọgwụ ahụ, a na-enweta mmetụta kachasị mgbe izu anọ gachara. Tupu ịmalite ọgwụgwọ, a ga-ebugharị onye ọrịa ahụ ka ọ bụrụ nri dị ala, nke a ga-ahụrịrị n'oge ọgwụgwọ ọgwụ.

Atoris dị n'ụdị mbadamba ya na atorvastatin na olu nke 10, 20 na 40 mg kwa mbadamba.

Ihe ngosi maka ojiji

Gịnị na-enyere Atoris aka? Kọwaa ọgwụ ahụ n'ọnọdụ ndị a:

  • maka ọgwụgwọ nke ndị ọrịa nwere isi (ụdị 2a na 2b) yana hyperlipidemia agwakọta.
  • A na-egosi nchịkwa nke ọgwụ maka ndị ọrịa nwere ezinụlọ hyzycholesterolemia na ezinụlọ nwere ụba: cholesterol n'ozuzu, obere lipoprotein cholesterol, triglyceride ma ọ bụ apolipoprotein B.

Ntụziaka maka iji Atoris, usoro onunu ogwu

A na -e oara ọgwụ ahụ ọnụ, n'agbanyeghị nri.

Usoro akwadoro ibido bụ 1 mbadamba Atoris 10 mg kwa ụbọchị. Dabere na ntuziaka ahụ, usoro ị ofụ ọgwụ ahụ si na 10 mg ruo 80 mg otu ugboro kwa ụbọchị, ma ahọpụtara na-eburu n'uche usoro mbụ nke LDL-C, ebumnuche ọgwụgwọ na mmetụta ọgwụgwọ nke onwe ya. Ọ bụ dibịa bekee na-elele otu a ga-esi nweta ọgwụ ahụ, na-eburu n'uche nsonaazụ nyocha ahụ na ọkwa mbụ nke cholesterol.

Na mbido ọgwụgwọ na / ma ọ bụ n'oge mmụba nke dose ahụ, ọ dị mkpa iji nyochaa ọdịnaya ụrọ plasma kwa izu 2-4 ma mezie ọnụọgụ ahụ dabere.

Na isi (heterozygous hereditary na polygenic) hypercholesterolemia (ụdị IIa) yana hyperlipidemia agwakọta (ụdị IIb), ọgwụgwọ na-amalite site na usoro ọgwụgwọ akwadoro, nke a na-abawanye mgbe izu anọ gachara dabere na nzaghachi onye ọrịa. Oke kachasị kwa ụbọchị bụ 80 mg.

Maka ndị ọrịa agadi na ndị ọrịa nwere ọrụ mkpali na-arụ ọrụ, a naghị achọ ndozi dose.

N'ime ndị ọrịa nwere ọrụ imeju na-egbu egbu, a na-enye ọgwụ ahụ iji nlezianya na-emetụta njikọ dị na mkpochapu ọgwụ na ahụ.

Nsonaazụ

Dịka ntuziaka maka ojiji esi mee, Atoris nwere ike sonyere nsonaazụ ndị a:

  • Site na psyche: ịda mba, ọgba aghara ụra, gụnyere ehighị ụra ehihie na abalị.
  • Site na usoro ahụ ji alụso ọrịa ọgụ: mmeghachi ahụ nfụkasị ahụ, anaphylaxis (gụnyere ụjọ anaphylactic).
  • Ọrịa metabolism: hyperglycemia, hypoglycemia, ibu ibu, anorexia, ọrịa shuga mellitus.
  • Site na usoro ịmụ nwa na mammary glands: dysfunction mmekọahụ, enweghi ike, gynecomastia.
  • Site na usoro ụjọ ahụ: isi ọwụwa, paresthesia, dizziness, hypesthesia, dysgeusia, amnesia, neuropathy akụkụ.
  • Site na sistem iku ume: ọrịa ngụgụ, ọnya na akpịrị, imi.
  • Ọrịa na ọrịa: nasopharyngitis, ọrịa urinary.
  • Site na sistemu ọbara yana sistem lymphatic: thrombocytopenia.
  • Site n'akụkụ akụkụ ahụ nke ọhụụ: ahụrụ ọhụhụ, ahụhụ ụzọ.
  • Site na usoro obi: okpo iku ume.
  • N’akụkụ akụkụ anụ ahụ na-anụ ihe: tinnitus, ọnwụ ịnụ ihe.
  • Site na nri diges: afọ ntachi, flatulence, dyspepsia, ọgbụgbọ, afọ ọsịsa, ọgbụgbọ, mgbu na elu na ala afọ, belching, pancreatitis.
  • Site na sistemu ịba ọcha n'anya: ịba ọcha n'anya, cholestasis, ọrịa imeju.
  • Site na anụ ahụ na anụ ahụ dị n'okpuru ala: urticaria, ọnya anụ ahụ, itching, alopecia, angioedema, bulmat dermatitis, gụnyere exriative erythema, Stevens-Johnson syndrome, necrolysis na-egbu egbu, na -akasị ọnya ọnya.
  • Site na usoro akwara: myalgia, ọrịa ogbu na nkwonkwo, mgbu aka, azụ mgbu, nkwonkwo azụ, mgbu azụ, mgbu olu, ike ọgwụgwụ, myopathy, myositis, rhabdomyolysis, tendonopathy (mgbe ụfọdụ ihe na-agbasi ike site na mgbatị anụ ahụ).
  • Ọrịa ndị a na-ahụkarị: malaise, asthenia, mgbu obi, oke ọgụ, ike ọgwụgwụ, ahụ ọkụ.

Ihe ngbanwe

Atoris na contraindicated na ndị a:

  • mmadu imegodi ihe ọgwụ di iche iche,
  • galactosemia,
  • malabsorption nke glucose galactose,
  • ụkọ lactose,
  • nnukwu akụrụ ọrịa,
  • ntụpọ akwara nke ọkpụkpụ,
  • tụụrụ ime
  • inye ara
  • afọ ruru 10.

Ekwesịrị ịkpachara anya na mmanya, ọrịa imeju. Otu a tinyekwara ndị ọrụ ọrụ ha metụtara ịkwọ ụgbọala na usoro dị mgbagwoju anya.

Dodoụbiga ya ókè

N'ihe banyere ịdoụbiga mmanya ókè, ekwesịrị ịgwọ ọrịa Symptomatic na nkwado nkwado. Ọ dị mkpa ijikwa ọrụ imeju yana ọrụ CPK n'ọbara. Ọkpụkpụ anụ ahụ adịghị arụ ọrụ. Enweghị ọgwụ mgbochi akọwapụtara.

Analogs Atoris, ọnụahịa dị na ahịa ọgwụ

Ọ bụrụ na ọ dị mkpa, enwere ike dochie Atoris na analog nke ihe dị n'ọrụ - ndị a bụ ọgwụ ọjọọ:

Mgbe ị na-ahọrọ analogues, ọ dị mkpa ịghọta na ntuziaka maka iji Atoris, ọnụahịa na nyocha nke ọgwụ nwere otu mmetụta emetụtaghị ya. Ọ dị mkpa ịnweta ndụmọdụ nke dọkịta na ịghara ime mgbanwe ọgwụ ọ bụla.

Na-echekwa na okpomọkụ agaghị akarị 25 Celsius. Ndụ shelf bụ afọ 2. N'ime ụlọ ahịa ọgwụ, ọgwụ na-ere ya.

Enwere nyocha dị iche iche banyere Atoris, ebe ọtụtụ na-ekwu na ọnụ ahịa ọgwụ dị elu ziri ezi site na ịdị mma ya na ntachi obi dị mma.

Achọpụtara na n’oge ọgwụgwọ, ekwesịrị ịgbaso ntuziaka dọkịta banyere nri na mmega ahụ, yana mgbe ị na-ahọrọ ma dozie ọgwụ ahụ, ekwesịrị ịbanye n’ogoproteins dị ala.

Dabere na ụfọdụ ndị ọrụ, ọgwụ ahụ enweghị mmetụta ọgwụgwọ kwesịrị ekwesị yana enweghị ndidi na-ezighi ezi, na-akpata mmeghachi omume ọjọọ.

Ihe atoris analogues dị ọnụ ala

Iji belata ọkwa nke lipids n'ọbara, ndị dọkịta na-eji ọgwụ dị iche iche, n'etiti Atoris na analogues na-ewu ewu. Ha na-achọ ibelata cholesterol ọbara, si otú a mee ka ọdịmma mmadụ n'ozuzu ya ka mma.

Banyere ọgwụ

A na-emepụta mbadamba nkume Atoris na Slovenia. Ọgwụ a bụ nke ụdị “akpụ akpụ” a na-enyekwa ya ndị ọrịa ka ha belata ogo nke lipoproteins dị ala (ihe na-enye nsogbu cholesterol) n’ahụ.

Atorvastatin bụ isi ihe eji agwọ ọgwụ. Site n'ime ka ọbara banye n'ime akwara, atorvastatin na - akwụsị njikọ nke ụmụ irighiri cholesterol site na mkpụrụ ndụ imeju.

N'ime usoro a, n'ahụ mmadụ na-amalite itinye aka nke lipoproteins nke banyeworo n'ọbara, na-enwe ntakịrị pasent nke njupụta.

N'ihi nke a, arụmọrụ nke Atoris na analogues ya, nke nwere ụdị ọrụ a na-arụ, na-abawanye.

Mkpochapu egbugbere ọnụ nke Atheis na-akpata anaghị eduga na njedebe nke ikpeazụ na mgbidi arịa ọbara. N'otu oge ahụ, atherosclerosis anaghị etolite etolite ọbara adịghị etolite. Ọ bụrụ na ischemia na-aga n’ihu n’ahụ mmadụ, iwere Atoris na akwara ndị ahụ na-eduga n’ịbelata ihe ize ndụ nke ịmalite ọrịa strok na nkụchi obi.

Formdị Atoris na usoro onyonyo ya na-egosi ị useụ ọgwụ dịka otu dibia bekee siri kwupụta.

Ọtụtụ mgbe, dabere na ọnọdụ ahụ dum na usoro akwara obi, dọkịta na-ekpebi usoro ọgwụgwọ dị mkpa iji mee ka ahụike ka mma.

Otutu oge, Atoris na analorọ ya bu ihe ndi edebere na ala, ebe nke a na-ebelata ohere nke ogba ojoo.

Atoris analogues nke na-esighi ike n'ịgwọ ọgwụ n'onwe ya ka ejirila na ahụike kemgbe ihe karịrị afọ iri. Nke a na-egosi na site na ọtụtụ nyocha dị mma nke ndị dọkịta na ndị ọrịa. Site na hypercholesterolemia, Atoris na analogues ya nwere ike belata cholesterol ka ọ bụrụ ọkwa dị mma maka obere oge, ebe ibelata ibu ahụ na obi.

Ruo ugbu a, ọtụtụ ndị Atoris analogues ejirila ndị dibịa belata cholesterol ọbara. Na Russia, na shelves nke pharmacies, a na-egosi ọgwụ ndị kwekọrọ na ọ bụghị naanị na mbubata, kamakwa n'ime ime ụlọ. Ihe ana-eme Atoris n’otu n’otu nwere udiri ya na udiri oru, ndi dibia gha aghaghi iburu n’uche tupu ogwu edee ya.

Rosuvastatin

Rosuvastatin bụ mbadamba ụrọ nke agba pink ma ọ bụ nke na-acha odo odo. Dị ka isi ihe na - arụ ọrụ bụ ụmụ irighiri rosuvastatin, nke ihe dị iche iche. Na mgbakwunye na ya, mbadamba nkume nwere:

  • magnesium stearate
  • eriri stachi
  • ụdị nke silicon dioxide,
  • ihe mgbochi hypromellose,
  • ncha pụrụ iche
  • triacetin
  • microcrystalline cellulose,
  • titanium dioxide.

Ihe eji arụ ọrụ nke mkpụrụedemede ndị ahụ akọwara bụ ihe eji arụ ọrụ nke enzymes ndị mmadụ n'otu n'otu na-arụ maka ịkpụpụta ụmụ irighiri mevalonate. Nke ikpeazụ, a na-agwakọta cholesterol.

Otu ọgwụ, nke Rosuvastatin bụ nke ya, na-akwụsị njikọ nke ụmụ irighiri ihe mevalonate.

Mgbe mmejuputara mmezu ya, a na-ewepụ ọgwụ ahụ n'ụdị na-agbanweghi n'ahụ ya na anụ ahụ.

E nyere ndị ọrịa nwere mkpụrụedemede ana –aeringụ dị ala, nke bụ rosuvastatin.

  • ụdị nke hypercholesterolemia,
  • hypertriglyceridemia,
  • ọdịdị homozygous (ezinụlọ) nke hypercholesterolemia.

Usoro onodu ogwu eji eme ihe mgbe ị na-ewere analog bụ nke dọkịta ji enyere ya aka mgbe ọ bụla iji belata nsogbu ị nwere ike ịkpalite ọrịa mgbochi atherosclerosis. A na-enyekarị Rosuvastatin ndị ọrịa oge agadi, ebe ọ bụ na n'oge a, lumens nke ọtụtụ arịa ha nwere dayameta kachasị nta, ebe ọ bụ na cholesterol jupụtara.

Obe a bu mbadamba pink nke nwere pink nwere ihe di n’ime ya. Ọ bụ ya na-arụ ọrụ nke nnukwu ọgwụ ọgwụ ahụ. Ntinye uche nke ihe na-arụ ọrụ mgbe ị na-ewere Krestor site na dọkịta, mgbe nyocha zuru oke.

Ọgwụ a dị irè maka hypercholesterolemia, yana maka hypertriglyceridemia.

Ọzọkwa, a na-eji ọgwụ ahụ agwọ ọrịa mellitus na-abụghị insulin na-akpata. Mbibi nke ọgwụ ahụ na-apụta na mkpụrụ ndụ imeju, ihe na-esochi ahụ sitere na ahụ.

Were analog kwesịrị iji obere mmiri. Edere ọtụtụ na usoro nhọpụta ndị dọkịta ka nyochachara nyocha pụrụ iche nke usoro ọbara nke onye ọrịa. Onwe-ogwu nke Krestor di ize ndu nye ahụ ike, ebe o nwere ike bute nsonaazụ ma a caseụbiga ya oke.

Cardiomagnyl

Cardiomagnyl bu ihe ozo nke anorọ nke Atoris. Ihe ndị nọ n'ọrụ bụ ụmụ irighiri acetylsalicylic acid nwere magnesium hydroxide. Mmụba na ọrụ 'cholesterol ọjọọ' n'ime ọbara ọbara na-egosi nhọpụta nke Cardiomagnyl site na dọkịta nye onye ọrịa!

Thisụ ọgwụ a na-eme ka o nwee ohere ịba uru nke thrombosis intravascular n’ime ahụ. Nke a mere mgbe:

  • ụdị ejighi angina pectoris,
  • ọrịa shuga,
  • oke ibu n’arụ
  • ọbara mgbali elu
  • infarction myocardial.

Cardiomagnyl bụ contraindicated na ndị mmadụ na-ata ahụhụ site na:

  • allergies na ọgwụ,
  • ọbara ọgbụgba n'ụbụrụ,
  • eriri afọ,
  • ụkọ ke ahu-K-vitamin,
  • ihe mgbu na ọnya ọgbụgba n'ime akụkụ akwara nri,
  • oke ogo siri ike gbasara akwara.

Anaghị anabata Cardiomagnyl ndị mmadụ na-ata ahụhụ na ntachi obi ha n'ahụ ụmụ irighiri Acetylsalicylic acid na magnesium hydroxide, yana n'oge afọ ime n'oge a na-ebu lactation.

Simvastatin

Atoris ma ọ bụ simvastatin dị irè karị? Simvastatin bụ ọgwụ hypoliplera nke nwere nnukwu ihe nke otu aha ahụ. Edere ọgwụ ọgwụ a maka ndị ọrịa na-arịa oke ọdịnaya nke sọks dị ka akwara dị n'ọbara.

N'ihi nke a, enweghị mkpokọta ogige ikuku na-egbu egbu na ahụ. Site n'ịba uru dị elu nke ọgwụ ahụ, ọgwụ ahụ nwere ọnụ ahịa a na-anakwere, nke na-eme ka ọ bụrụ ndị a ma ama n'etiti ndị bi. Mmepe nke myopathy mmadụ bụ ihe nnọchianya iji kwụsị ị thisụ ọgwụ a.

Atoris ma ọ bụ Atorvastatin: nke ka mma? Tupu ịhọrọ atụ nke Atoris, ị kwesịrị ịgakwuru dọkịta gị, mgbe nyochachara anụ ahụ zuru ezu, ga-enwe ike ịde ọgwụ ọfụma na nke dị mma maka onye ọrịa.

Anyị na-akwado ya! Maka ọgwụgwọ na mgbochi nke ọrịa JOINTS NA SPINE, ndị na-agụ akwụkwọ anyị na-eji usoro nke ọgwụgwọ ngwa ngwa na-enweghị ịwa ahụ nke ndị isi ọrịa Russia na-atụ aro, bụ ndị kpebiri na-emegide mmebi iwu ọgwụ ma wepụta ọgwụ na-egosi n'ezie! Anyị matara usoro a ma kpebie itinye uche gị na ya.

Atoris: ntuziaka maka ojiji, analogues, ọnụahịa, nyocha

Atoris bụ otu aha azụmaahịa maka atorvastatin nke ụlọ ọrụ Slovenian Krka mepụtara. N'ime usoro ọmụmụ ndị ọzọ, ọgwụ a pụtara nke ọma.

E nyere Atoris ka cholesterol dị ala, "lipoproteins" na-emerụ ahụ, triglycerides, yana iwelie ịta "ezigbo lipoproteins.

Ntụziaka ahụ gosipụtara na ndị lekwasịrị anya na ọgwụ Atoris bụ ndị mmadụ na-arịa ọrịa hypercholesterolemia, ọrịa obi obi (CHD), na ọrịa shuga mellitus.

Ngwakọta, ụdị ntọhapụ

Atoris bụ mbadamba nkume nwere miligram 10, 20, 30, 60, ma ọ bụ 80 nke ihe arụ ọrụ. Gburugburu, convex, na-acha ọcha. Na mmejọ - ok, ọcha.

Ihe arụ ọrụ nke Atoris bụ calcium atorvastatin. Na mgbakwunye na ya, ihe mejupụtara ọgwụ ahụ bụ: povidone, sodium lauryl sulfate, calcium carbonate, cellulose, lactose monohydrate, croscarmellose, magnesium stearate. A na-etinye mbadamba ọ bụla na Opadry 2.

Atoris: ngosipụta maka ojiji

Tupu ị takingụ ọgwụ ahụ, a na-ebugharị onye ọrịa ahụ na nri nke na-eme ka mkpokọta cholesterol, ọbara LDL belata. Ekwesịrị ịhụ ya n'oge usoro ọgwụgwọ. Ileghara nri anya riri ma obu mebie oru oma ọgwụgwọ atorvastatin.

Dịka ntuziaka ahụ si dị, a na-eji mbadamba nkume Atoris agwọ:

  • homo-, heterozygous ezinụlọ na hypercholesterolemia na-abụghị nke ezinụlọ.
  • jikọtara hyperlipidemia,
  • dysbetalipoproteinemia,
  • Ezigbo nsogbu hypertriglyceridemia.

Atoris ka edekwara maka igbochi oria obi agha. N'ihi mgbochi nke atherogenic nke ọgwụ:

  • na-eme ka mmadụ ghara ibute ọrịa obi,
  • na-ebelata ohere nke nkụchi obi, ọrịa iku ume,
  • na-egbochi mwakpo angina,
  • belata ọnụ ọgụgụ ndị ọrịa chọrọ ịwa ahụ.

Ofzọ nke ngwa, usoro onunu ogwu

A na-ewere mbadamba Ator otu ugboro / ụbọchị tupu ụra, tupu, mgbe ọ gasịrị ma ọ bụ jiri nri. Ọ bụ ihe amamihe dị na ya ị takeụ ọgwụ ahụ n'otu oge.

Gịnị kpatara o ji dị mkpa iburu Atoris na mgbede? N'abalị, imeju na - agbakọta ihe kacha cholesterol. Ọ bụrụ n’ichefu ịillụ ọgwụ, mee ya ozugbo enwere ike.

Ghafee otu oge atọrọ ma ọ bụrụ na erughị elekere iri na abụọ ka ọnwa na-abịa. N'otu oge, ekwesighi ịba ụba nke ọgwụ a.

The recommendedụ ọgwụ a tụrụ aro ya bụ 10-80 mg. Mgbe ị na-ahọrọ usoro onoris nke Atoris, cholesterol mbụ, LDL, ọnụnọ nke nsogbu concomitant, na iji ọgwụ ndị ọzọ na-eburu n'uche.

Ọgwụgwọ bidoro na obere usoro ọgwụ a (10-20 mg). Mgbe izu anọ gachara, dọkịta ahụ nyochachara mgbanwe nke mgbanwe na cholesterol, lipoproteins. Ọ bụrụ na arụpụtaghị mmetụta achọrọ, a na-abawanye dose nke Atoris. N'ihe cholesterol dị ala, a na-enye mbadamba ihe nwere ike itinye ihe n'ọrụ.

Iji dozie cholesterol, a na-enye ndị ọrịa na-ewere erythromycin, clarithromycin, lopinavir, ritonavir, Atoris na dose nke na-erughị 20 mg.

N'oge ọgwụgwọ, ọ dị mkpa ijikwa ọkwa cholesterol, LDL, VLDL, triglycerides, imeju, akụrụ, CC. Nke a na - enyere aka ịtụle mmeghachi omume nke anụ ahụ maka ojiji nke Atoris, yana ịchọpụta mmepe nke nsonaazụ na oge.

Mmekorita

N’otu oge eji mbadamba nkume Atoris nke nwere ufodu ogwu n’enweghi nsogbu site na ihe ojoo di ya ma obu ibelata idi nma otu n’ime ha.

Edeghi ọgwụ a maka ndị na-a :ụ ọgwụ:

  • ọgwụ antifungal nke otu azole,
  • ụfọdụ ọgwụ nje (cyclosporine, telithromycin),
  • gemfibrozil
  • Ihe nchedo nje HIV (ritonavir, lopinavir),
  • fusidic acid
  • na-a juiceụ mkpụrụ osisi grape.

Medicationsfọdụ ọgwụ, mgbe ejikọtara ya na Atoris, chọrọ ndozi usoro onunu ogwu. Ndepụta ha dị na ngalaba "hodzọ nke ngwa na usoro onunu ogwu."

Ahapụ Gị Ikwu