Mbadamba ụrọ nke Ovencor: ngosipụta maka ojiji, ọnụahịa na analogues

Ariescore (ọgwụ) Rating: 9

Emeputa: Ozone (Russia)
Mwepụta Mwepụta:

  • Tab. 10 mg, pcs iri abụọ., Ọnụ ego sitere na 372 rubles
  • Tab. 20 mg, pcs iri abụọ., Ọnụ ego site na 510 rubles
Ọnụ ego dị elu n’ahịa ọgwụ dị n'ịntanetị
Ntụziaka maka ojiji

A na-emepụta ọgwụ ahụ na Russia, ezubere maka ọgwụgwọ nke ọrịa nke usoro obi. Ihe dị n'ọrụ bụ simvastatin na ọnụọgụ 10 ma ọ bụ 20 mg kwa mbadamba. Contraindicated n'okpuru afọ 18 afọ.

Analogs nke ọgwụ Ariescor

Ihe analogue dị ọnụ ala site na 313 rubles.

Emeputa: Vertex (Russia)
Mwepụta Mwepụta:

  • Mbadamba ụrọ 10 mg, 15 PC., Ọnụ sitere na 59 rubles
  • Mbadamba 10 mg, 30 PC., Ọnụ ego site na 62 rubles
Ọnụ ego Simvastatin n'ụlọ ahịa ọgwụ dị n'ịntanetị
Ntụziaka maka ojiji

Simvastatin bụ ọgwụ na-egbusi ike nke mmepụta Russian. Ọ dị n'ụdị mbadamba nkume ma nweekwa otu ihe eji arụ ọrụ n'ime usoro nke 10 ruo 40 mg. Egosiputa ya maka ọgwụgwọ nke ọrịa nke ọrịa obi.

Ihe analogue dị ọnụ ala site na 173 rubles.

Emeputa: Krka (Slovenia)
Mwepụta Mwepụta:

  • Mbadamba 20 mg, pcs iri na anọ., Ọnụ ego site na 199 rubles
  • Mbadamba 10 mg, 28 PC., Ọnụahịa site na 289 rubles
Ọnụ ahịa Vasilip na ụlọ ahịa ọgwụ dị n'ịntanetị
Ntụziaka maka ojiji

Onye ọzọ ga-aba uru na Slovenian otu ụdị ntọhapụ yana otu ihe bekee na-arụ ọrụ. Isi ihe ngosi maka ojiji: hypercholesterolemia bụ isi ma ọ bụ ọrịa dyslipidemia, mbelata ọnwụ nke obi na ọrịa na ndị ọrịa nwere ngosipụta nke akwara nke ọrịa obi atherosclerotic ma ọ bụ ọrịa shuga mellitus. Enwere contraindications.

Ihe analogue dị ọnụ ala site na 265 rubles.

Emeputa: Gideon Richter (Romania)
Mwepụta Mwepụta:

  • Tab. 10 mg, pcs iri na anọ., Ọnụ ego site na 107 rubles
  • Tab. 10 mg, 28 PC., Ọnụ sitere na 202 rubles
Ọnụ ego Simvastol na ụlọ ahịa ọgwụ dị n'ịntanetị
Ntụziaka maka ojiji

Simvastol bụ analog nke mmepụta Romania. Odikwa n’ime kaadiboodu nke 14 na mbadamba 28. Ihe na-arụ ọrụ bụ otu ihe ahụ ebe a, yabụ ntuziaka maka ojiji nwere naanị obere ọdịiche. Tupu ịmalite ọgwụgwọ, anyị na-akwadosi ike ịkpọ dọkịta.

Mwepụta wepụtara ya na ihe mejupụtara

Usoro onunu ogwu Ovenkor weputara - mbadamba mkpuchi nwere: acha ọcha, biconvex gbara okirikiri (10 ma obu 30) Na blisters, n’ime igbe kaadi 10, 20, 40, 60, 80 na 100, 10, 14, 20, 28, 30, 40, 50 ma ọ bụ 100 PC. Na polymer containers, na a kaadiboodu ukwuu 1 akpa).

Ngwakọta 1 mbadamba:

  • ihe na-arụ ọrụ: simvastatin - 10 ma ọ bụ 20 mg,
  • ihe inyeaka: polyethylene glycol-4000, talc, titanium dioxide, castor, butyl hydroxyanisole, microcrystalline cellulose, ascorbic acid, lactose, citric acid, ọka na pregelatinized starches, magnesium stearate, hydroxypropyl methylcellulose.

Mlọ ọgwụ

Ọgwụ sitere na otu nke statins, nwere mmetụta dị ala, belata HMG-CoA reductase. Ọdịdị ya emechiri emechi lactone mgbanaka, nke a na - eme mmiri n’ime ahụ mmadụ, ya bụ, ọ bụ prodrug.

Lactone mgbanaka statins nwere mmekọrịta maka enzyme HMG-CoA reductasen'ihi nke ọ na asọmpi na-ekekọta akụkụ nke onye na-anabata ya coenzyme Aebe enzyme a na-akwado.

Akụkụ nke statin molecule na-etinye aka na ntụgharị hydroxymethylglutarate n'ime mevalonatenke metụtara ngwaahịa nke etiti ana - eme ihe na - eme ihe cholesterol. Usoro ndị a na-akpata ọtụtụ mmeghachi omume, n'ihi nke ọdịnaya intracellular dị cholesterol belata catabolis cholesterol cholesterol LDL. Mmetụta ịdị ala nke ọgwụ bụ n'ihi mbelata cholesterol na-ebelata n'ihi cholesterol LDL. N'otu oge ahụ, mbelata nke ọkwa nke LDL dose-dabere na bụ exponential.

Statins anaghị emetụta catabolism na njikọ nke abụba n'efu, yabụ ha na-emetụta ọkwa nke TG udiozi (nke abuo). Dabere na ọmụmụ, ọgwụ na-ewelite ọkwa nke Cholesterol HDL ruru 14%. Na mgbakwunye na mmetụta lipid, ọgwụ ahụ nwere mmetụta dị mma na mgbidi vaskụla n'oge nsị nke endothelial (akara ngosipụta nke ihe ngosipụta mbụ nke atherosclerosis), na-ahụ maka ihe ndị metụtara ọbara na ọbara, ma nwee mmetụta antiproliferative na antioxidant. Ọgwụ yana iji ọgwụ a sobelata ugboro ugboro ọrịa obi.

Mlọ ọgwụ

Simvastatin nwere mmịpụta dị elu. Oke itinye uche na plasma ọbara mgbe ịbanyechara mmadụ bụ emesịrị ihe dị ka awa 1.3-2.4, mgbe awa 12 ọ jiri 90% belata. Nkwurịta okwu na protein ndị na-edozi ahụ bụ ihe dị ka 95%.

O nwere nsonaazụ nke akụkụ mbụ site na imeju: hydrolysis na usoro nke beta-hydroxyacid dị n'ọrụ, a chọpụtakwara metabolites ndị ọzọ na-arụ ọrụ na-adịghị arụ ọrụ.

Mwepu ọkara ndụ nke metabolites nọ n'ọrụ bụ awa 1.9.

Emere ya tumadi n'ụdị metabolites na feces (60%). N’ụdị arụ ọrụ, ihe dị ka 10-15% ka akụrụ wepụtara.

Ihe ngosi maka ojiji

  • hypercholesterolemia: hypercholesterolemia nke mbụ (ụdị IIa na IIb) na ndị ọrịa nwere oke ihe na-etolite akwara na atherosclerosis n'ihe banyere usoro ọgwụgwọ nri na-adịghị mma na cholesterol dị ala na usoro ndị ọzọ na-adịghị ọgwụ (oke ibu na ọrụ anụ ahụ), ngwakọta nke hypercholesterolemia na hypertriglyceridemia, nke na-anaghị edozi n'ụzọ pụrụ iche. mmega ahụ,
  • IHD (ọrịa obi): iji gbochie infarction myocardial, belata ihe mgbawa obi (ọrịa strok ma ọ bụ ọgụ azụ), ọnwụ, usoro ịmụgharị, yana iji belata oganihu akwara arteriosclerosis.

Ihe ngbanwe

  • ọrịa imeju na-arụ ọrụ na-arụ ọrụ, mmụba na-abawanye na ọrụ nke enzymes nke imeju amataghị,
  • porfria
  • myopathy
  • afọ ruo afọ 18
  • ime na lactation,
  • nnabata onwe onye maka ọgwụ a, yana ọgwụ ọgwụ statin ndị ọzọ (HMG-CoA reductase inhibitors) na akụkọ ntolite.

A na-ahọpụtara onye nlekọta (Ovenkor n'okpuru nlekọta ahụike):

  • ị .ụbiga mmanya ókè
  • hypotension artital, nnukwu ọrịa na-efe efe, ọrịa endocrine / metabolic na-adịghị ala ala, mmiri na-arịa mmiri elektrọnik, mmerụ ahụ, ihe ịwa ahụ (gụnyere eze) ma ọ bụ ọnọdụ ndị ọzọ enwere ike inwe mmepe nke nnukwu gbasara akụrụ,
  • ọnọdụ mgbe ebugharị akụkụ ahụ n'oge ọgwụgwọ immunosuppressant (ejikọtara ya na oke ihe ize ndụ nke ọdịda akụrụ na rhabdomyolysis),
  • Akwụkwụ na-adọ
  • mbelata / uda olu nke okpukpu ọkpụkpụ akwara nke mmalite amaghi.

Ntụziaka maka iji Ovenkor: usoro na usoro onunu ogwu

A na-ewere ọnụ nye Ovencor ugboro 1 n'ụbọchị na mgbede, jiri mmiri dị ukwuu sachaa ya. Oge ị takingụ ọgwụ agaghị ejikọta ya na iri nri.

Tupu ịmalite Ovenkor, a na-enye onye ọrịa iwu usoro hypocholesterol kwesịrị ekwesị, nke a ga-agbaso n'oge ọ bụla ọgwụgwọ.

Na hypercholesterolemia, ị dailyụ ọgwụ kwa ụbọchị dịgasị iche n'etiti 1080 mg.

Usoro akwadoro ịmalite hypercholesterolemia bụ 10 mg. Oke - 80 mg kwa ụbọchị. Ekwesịrị ime mgbanwe (nhọrọ) nke dose ahụ na etiti oge izu anọ. N'ọnọdụ ka ukwuu, a na-ahụ nsonaazụ kachasị mma mgbe ị na-a takingụ ọgwụ na ọgwụ kwa ụbọchị nke ruru 20 mg.

Site na hyzycholesterolemia homozygous, a na-enyekarị Ovencor ọgwụ na 40 mg na 1 mg ma ọ bụ 80 mg na usoro 3 (20 mg n'ụtụtụ na n'ehihie, 40 mg na mgbede).

Ngwọta dị irè nke Ovenkor maka ọrịa obi na -akpata ma ọ bụ ọnụnọ nke ihe dị ukwuu nke mmepe ya bụ 20-40 mg kwa ụbọchị. Na mbido usoro ọgwụgwọ, a na-enyekarị ọgwụ 20 mg, enwere ike ịbawanye dose ahụ na ezumike nke izu anọ. Mgbe ọdịnaya LDL erughị 75 mg / dl (1.94 mmol / L) yana cholesterol zuru ezu erughị 140 mg / dl (3.6 mmol / L), a na-ebelata ọgwụ ahụ.

N'ihe dịkarị nke 10 mg, Ovencor depụtara ihe na-erughị 30 ml / min na ndị ọrịa nwere ọdịda akwara na-adịghị ala ala (CRF) (creatinine nwechara) ma ọ bụ ọgwụgwọ ejikọtara ya na cyclosporine, danazole, gemfibrozil ma ọ bụ fibrates ndị ọzọ (ma e wezụga fenofibrate), niacin na lipid wedates doses ( ihe ruru 1000 mg kwa ụbọchị). Iji otu oge eji amiodarone ma ọ bụ verapamil, ọgwụ kwa ụbọchị nke Ovenor ekwesịghị gafere 20 mg.

Nsonaazụ

  • Usoro nri: afọ mgbu, afọ ntachi / afọ ọsịsa, flatulence, ọgbụgbọ, pancreatitis, ịba ọcha n'anya, vomiting, ụba ọrụ nke enzymes imeju, alkaline phosphatase na CPK (creatine phosphokinase),
  • akwara anụ ahụ na sistem ụjọ: isi ọwụwa, ọrịa asthenic, neuropathy ihu, ọgbụgbọ, ehighị ụra nke ọma, paresthesias, akwara mgbu, imebi ihe mmetụta dị ụtọ, ọhụhụ ụzọ,
  • immunopathological na mmeghachi omume nfụkasị: ọkụ na-ekpo ọkụ, eosinophilia, hyperemia nke anụ ahụ, ogbu na nkwonkwo, vasculitis, angioedema, polymyalgia rheumatism, thrombocytopenia, mụbara ESR, ọgwụ lupus-reversable syndrome dị ka ọrịa, ahụ ọkụ, urticaria, foto, mkpụmkpụ ume,
  • Ọrịa akpọnwụ anụ: na - adịkarịghị - dermatomyositis, ọnya anụ ahụ, alopecia, itching,
  • sistem mọzụlụ: adịghị ike, myopathy, olu mgbu, myalgia, adịkarịghị - rhabdomyolysis,
  • mmeghachi omume ndị ọzọ: palpitations, anaemia, nwere ikike belatara, nnukwu akụrụ gbasara ọdịda.

Dodoụbiga ya ókè

Onweghi ihe akara doro anya nke oke oke nke oke Ovenkor (a maara ihe banyere ị takingụ ọgwụ ahụ n ’ọgwụ nke 450 mg).

Usoro ọgwụgwọ: usoro nke iji belata nnabata nke ihe ahụ (itinye vomiting, na-ewere unyi na-arụ ọrụ), ọgwụgwọ Symptomatic n'okpuru nchịkwa gbasara akụrụ na ọrụ ịba ọcha n'anya, na ọkwa CPK serum.

N'ihe banyere mmepe nke myopathy na rhabdomyolysis na nnukwu gbasara akụrụ ọdịda (mmebi adịghị ụkọ, mana enwere ike ịda n'ụdị siri ike), a na-akwụsị Ovenkor ozugbo, a na-egosipụta nchịkwa nke diuretic na sodium bicarbonate (site na ntinye intravenous infusion). Ọ bụrụ na ọ dị mkpa, a na-awa ahụ.

Rhabdomyolysis nwere ike ibute hyperkalemia, nke a na-ewepụ site na nchịkwa intravenous nke calcium chloride ma ọ bụ glucose glucose, mgbakwunye glucose na insulin, ndị na-agbanye ọgwụ ion, ma ọ bụ, n'ọnọdụ ndị siri ike, site na hemodialysis.

Ntụziaka pụrụ iche

Na nmalite ọgwụgwọ, enwere ike ịbawanye nwa oge na ọkwa nke enzymes imeju.

Tupu ịkọwa ọgwụ ahụ ma na-eme n'ọdịnihu, a ga-eduzi ọmụmụ banyere ọrụ hepatic. Ugboro ole a na-enyocha ọrụ nke enzymes hepatic: ọnwa atọ mbụ - izu isii ọ bụla, mgbe ahụ n'ime afọ mbụ fọdụrụ - oge 1 na ọnwa abụọ, n'ọdịnihu - oge 1 na ọnwa isii. A na-ejikwa nnwale na-arụ ọrụ iji chọpụta ọrụ imeju na iji usoro ịba ụba. Ọ bụrụ na ọnụọgụ ahụ na-abawanye 80 mg kwa ụbọchị, njikwa kwesịrị ịme otu ugboro kwa ọnwa atọ. A kwụsịrị Ovenkor n'ihe banyere mmụba na-abawanye na ọrụ transaminase (ugboro atọ ma e jiri ya tụnyere ọkwa mbụ).

N'oge afọ ime, mwepu nke ọgwụ na-akụda Lipid na nsonaazụ nke ọgwụgwọ ogologo oge nke hypercholesterolemia enweghị mmetụta pụtara ìhè.

Aremụ nwanyị nọ n'afọ ndụ ịmụ nwa na-adịghị eji ọgwụ mgbochi eme ihe a naghị akwado ị takeụ Ovenkor.

Site na ọrụ thyroid na-ebelata (hypothyroidism) ma ọ bụ ọnụnọ nke ọrịa ụfọdụ akụrụ (ọrịa nephrotic syndrome) na mmụba nke cholesterol, ọrịa mbu ahụ kwesịrị ibu ụzọ gwọọ ya.

Ceptionnabata Ovenkor nwere ike iduga mmepe nke myopathy na ihe sochirinụ nke rhabdomyolysis na ọdịda akụrụ.

N'ọnọdụ mgbu mgbu, akwara olu, adịghị ike ma ọ bụ enweghị ike, ị kwesịrị ịkpọtụrụ dọkịta, ọkachasị ma ọ bụrụ na ọnya na ọnya na-arịa ọrịa ndị a. Umche / na-achọpụta myopathy, ọgwụgwọ akwụsịla.

Iji chọpụta ọrịa nke myopathy, a na-atụ aro ịlele ọnụahịa KFK mgbe niile. Na nchọpụta ọdịiche dị iche iche nke ihe mgbu n’azụ sternum, ị takingụ ọgwụ ahụ kwesịrị ịtụle.

Aries dị mma n'ụdị monotherapy ma jikọta ya na ndị na - esote bile acid.

Dọkịta na-ekpebi oge ọgwụgwọ dị iche iche.

Ime na lactation

Dabere na ntuziaka ndị ahụ, contraindicated na ụmụ nwanyị dị na Ovenkor n'oge afọ ime / lactation.

Enwere obere ihe akaebe banyere mmepe nke ara na ụmụ amụrụ ọhụrụ ndị nne ya tookụrụ ọgwụ ahụ. Womenmụ nwanyị nke afọ ịmụ nwa na-ewere simvastatin kwesịrị iji usoro mgbochi. Mgbe ime dị, Ovenkor na-akagbu ngwa ngwa.

Mkparịta ụka ọgwụ ọjọọ

  • erythromycin, immunosuppressants, telithromycin, clarithromycin, cytostatics, antifungal jami (ketoconazole, itraconazole), nefazodone, fibrates, nicotinic acid in a high doses, HIV proseres inhibitors: amụba ihe ize ndụ nke myopathy,
  • danazol, cyclosporine, gemfibrozil na ndị ọzọ fibrates (ewezuga fenofibrate), niacin, amiodarone, verapamil, diltiazem: ihe egwu nke myopathy / rhabdomyolysis,
  • anticoagulants na-egbu egbu (fenprocoumone, warfarin): ihe ize ndụ nke ọbara ọgbụgba, nlekota ọbara coagulability tupu ọgwụgwọ yana mgbe ezuru oge mmalite ọgwụgwọ,
  • digoxin: abawanye na ọkwa plasma ya,
  • colestipol, colestyramine: belatara bioavailability (ị ga - ewere Ovencor awa anọ mgbe ị theseụchara ọgwụ ndị a, ebe a na - achọpụta mmepe nke mmetụ ahụ),
  • ihe ọ juiceụụ mkpụrụ osisi (ihe karịrị 1000 ml kwa ụbọchị): mmụba dị ukwuu na ọkwa nke ọrụ inhibitory megide HMG-CoA reductase na plasma ọbara (a ga-ezere mkpokọta).

Ihe atụ nke Ovenkor bụ: Simvalimite, Sinkard, Zorstat, Simvastatin, Holvasim, Simgal, Zokor, Simvor, Simlo, Vasilip, Simvastol.

Nkọwapụta ọgwụ ọjọọ

Aries - Onye na - ahụ maka hypolipPs sitere na otu nke statins, onye na - egbochi HMG-CoA reductase. Ọ bụ prodrug, n'ihi na o nwere mgbanaka lactone mechiri emechi, na-agbanye mmiri mgbe ọ batachara ahụ.

Ọdịdị nke statin lactone ring dị ka nke akụkụ nke enzyme HMG-CoA. Dabere na ụkpụrụ ịsọ mpi ịkwa iko, mpekere statin na - ejikọ akụkụ ahụ Coenzyme A receptor ebe enzyme a na - etinye. Akụkụ ọzọ nke statin molecule na-egbochi ntụgharị nke hydroxymethylglutarate na mevalonate, ihe na-etiti na njikọ nke ụmụ irighiri cholesterol. Mgbochi ọrụ HMG-CoA reductase na-eduga n'usoro nke mmeghachi omume nke usoro, na-ebute mbelata ọdịnaya choralerol intracellular yana mmụba ụgwọ ọrụ nke ndị na-anabata LDL ma, ya mere, catabolism nke LDL cholesterol (Xc) na-akpata ike ngwa ngwa.

A na - ejikọta mmetụta hypolipPs nke statins na mbelata ọkwa nke cholesterol zuru oke n'ihi cholesterol LDL. Mbelata nke LDL bụ ihe dabere na nkwụchi ọnweghị akara, kama ọ dị mkpa.

Statins anaghị emetụta ọrụ nke lipoprotein na hepatic lipases, anaghị emetụta njikọ na catabolism nke ọdụdụ abụba n'efu, yabụ, mmetụta ha na ọkwa TG bụ nke abụọ na enweghị isi site na nsonaazụ ha bụ isi dị ala nke LDL-C dị ala. Mbelata nke ọkwa TG n'oge na -elezi anụ ahụ pụtara na ngosipụta nke ndị na-anabata ihe (apo E) ndị na-enweta hepatocytes metụtara catabolism nke STD, nke nwere ihe dịka 30% TG.

Dabere na ọmụmụ a na-achịkwa, simvastatin na-abawanye ọkwa HDL-C ruo 14%.

Na mgbakwunye na mmetụta mmetụ egbugbere ọnụ, statins nwere ezigbo mmetụta endothelial dysfunction (kpọmkwem akara nke atherosclerosis n'oge), na mgbidi vaskụla, steeti atheroma, melite akụrụngwa ọbara, nwere antioxidant, Njirimara antiproliferative. Enwere ihe akaebe na simvastatin na-emezi ọrụ endothelial mgbe ụbọchị 30 nke ọgwụgwọ gasịrị.

Ojiji simvastatin tinyere mbelata ugboro ugboro nke ọrịa obi, na agbanyeghị ọkwa mbu nke LDL-C.

Ndepụta nke analogues


Mpempe mwepụta (site na ama ama)Ọnụahịa, tee.
Aries
Mbadamba 20 mg, 30 PC.476
Avestatin
Na-eme ihe
Atherostat
Tab. 0,02 Nke 30 (AVVA RUS OJSC / Sti - Med - Sorb OJSC (Russia)232
Tb PO 0.02 Nke 30 (ABVA RUS OJSC / Sti - Med - Sorb OJSC (Russia)232
Vasilip
Tab 10mg N28 Vector (KRKA, dd. Ebe ọhụrụ / mkpọ. Vector (Russia)329.60
Tab 20mg N28 Vector (KRKA, dd. Ebe ọhụrụ / mkpọ. Vector (Russia)458.20
Tab 40mg N28 (KRKA - Rus LLC (Russia)628.20
Vero-Simvastatin
Zovatin
Zokor
10mg Nke 28 tab (Merck Sharp na Dome, UK. (England)176
Zokor Forte
40mg Nke 14 tab (Merck Sharp na Dome, UK. (England)458
Tab 40mg N14 (Merck Sharp na Dome, UK. (England)519.90
Zorstat
SIMVAHEXAL
Tab 20mg N30 (Hexal AG (Germany)287.10
Tab 10mg N30 (Hexal AG (Germany)319.10
Tab 40mg N30 (Hexal AG (Germany)484.70
Simvakard
Tab 20mg N28 (ZENTIVA a.s. Czech Republic (Czech Republic)172
Tab 10mg N28 (ZENTIVA a.s. Czech Republic (Czech Republic)218.80
10mg Nke 28 tab (Zentiva k.s. (Czech Republic)242
Simvacol
Simvalimite
Simvastatin
10mg Nke 30 tab p / pl. (Borisovsky ZMP OJSC (Belarus)38.60
20mg Nke 30 tab p / pl.o (Borisovsky ZMP OJSC (Belarus)47.50
Tab 10mg N30 Alsi (Alsi Pharma ZAO (Russia)53.70
Tab p / pl. Ihe dị ka 20mg N30 Alsi (Alsi Pharma ZAO (Russia)54.50
20mg Nke 30 tab p / pl.o AVVA RUS (AVVA RUS OJSC (Russia)68.30
10mg Nke 30 tab p / pl.o (Ozone LLC (Russia))89.10
20mg Nke 30 tab p / pl.o (Ozone LLC (Russia))113.80
Tab 20mg N30 (Verteks ZAO (Russia)147.60
Tab 10mg N30 (Verteks ZAO (Russia)207.30
Tab 20mg N20 (Hemofarm A.D. (Serbia)257.30
Simvastatin alkaloid
10mg Nke 28 tab p / pl. (Alkaloid AO (Macedonia)59.80
Simvastatin Zentiva
10mg Nke 28 tab (Zentiva k.s. (Czech Republic)259.90
20mg Nke 28 tab (Zentiva k.s. (Czech Republic)335
40mg Nke 28 tab p / pl. (Zentiva k.s. (Czech Republic)498.70
Simvastatin Pfizer
Simvastatin Sanofi
Simvastatin * (simvastatin *)
Simvastatin-ALSI
Simvastatin-SZ
Mbadamba 40 mg, 30 PC. (Northern Star, Russia)91
Simvastatin-teva
Simvastatin-ferein
Simvastatin-Chaikafarma
Simvastatin granules
Simvastol
Tab 10mg N28 (Gideon Richter OJSC (Hungary)197.10
Simvor
Tab po 40mg Nke 30 (Ranbaxi Laboratories Limited (India)60.10
Tab po 20mg N30 (Ranbaxi Laboratories Limited (India)282
Simgal
Tab 10mg N28 (Aivex Pharmaceuticals s.r.o. (Czech Republic)287
40mg Nke 84 tab (Teva Czech Enterprises s.r.r.o. (Czech Republic)304.40
10mg Nke 28 tab (Teva Czech Enterprises s.r.o. (Czech Republic)321.50
20mg Nke 28 tab p / pl. (Teva Czech Enterprises s.r.r.o (Czech Republic)410
10mg Nke 84 tab p / pl. (Teva Czech Enterprises s.r.r.o (Czech Republic)609.90
40mg Nke 28 tab p / pl. (Teva Czech Enterprises s.r.r.o (Czech Republic)678
20mg Nke 84 tab (Teva Czech Enterprises s.r.o. (Czech Republic)870
Tab 40mg N84 (Aivex Pharmaceuticals s.r.o. (Czech Republic)1505
Simlo
Tab 10mg Nke 28 (Ipka Laboratories Limited (India)202.90
Tab 20mg N28 (Ipka Laboratories Limited (India)293.60
Simplacor
Kaadi
Holvasim

Otu onye ọbịa kwuru na ụbọchị ọ ga-agwụ

Ogologo oge ole Ovencor na-eche na onye ọrịa ahụ na-akawanye mma?
Ndị sonyere na nyocha ahụ n'ọtụtụ oge ka ụbọchị otu ụbọchị nwetachara nkwalite. Ma nke a nwere ike ọ gaghị adakọ oge ị ga - emeziwanye. Gwa dọkịta gị ogologo oge ịchọrọ ị thisụ ọgwụ a. Tebụl dị n'okpuru ebe a na-egosi nsonaazụ nke nyocha na mmalite nke ihe dị irè.
Ndị otu%
1 ikp1

Otu onye ọbịa kọrọ banyere oge ọhụhụ

Kedu oge dị mma iji were Ovenkor: na afọ na-enweghị ihe ọ bụla, tupu ya, ma ọ bụ mgbe nri?
Ndị na-eme ihe ntanetị na-akọkarị ka ị takingụ ọgwụ a na afọ efu. Agbanyeghị, dọkịta nwere ike ịkwado oge ọzọ. Akuko ahụ gosipụtara mgbe ndị ọrịa ndị ọzọ gbara ajụjụ ọnụ na-a theụ ọgwụ.
Ndị otu%
Na afọ efu1

Ndị ọbịa iri na asaa kọtụrụ afọ ole ha dị

Ndị otu%
> 60 afọ12
70.6%
Afọ 46-60317.6%
30-45 afọ2

Ntụziaka gọọmentị maka ojiji

(Simvastatin) Nọmba ndebanye: LSR-002033/08
Aha ahia: Aries

Aha International nonproprietary: Simvastatin * (simvastatin *)

Mpempe usoro onunu ogwu: mbadamba ihe mkpuchi
Ngwakọta: 1 mbadamba ihe mkpuchi fim nwere
ike ọrụ: Ariescore - 10 mg ma ọ bụ 20 mg,
ndị na-ebu ụzọ: microcrystalline cellulose, lactose (shuga mmiri ara ehi), ahịhịa pregelatinized (stachi 1500), colloidal silicon dioxide (aerosil), ascorbic acid, butylhydroxyanisole, stearic acid, magnesium stearate, opadry II (polyvinyl mmanya, polyglycol ojii, gol iron) talc, iron dye oxide edo edo, iron dye oxide red, titanium dioxide).
Nkọwa: mbadamba biconvex gbara okirikiri, ihe mkpuchi na-acha odo odo, site na aja aja ruo na agba aja aja nke nwere agba pink.
Ndị na-ere ọgwụ: onye nnọchi anya belata, HMG-CoA reductase inhibitor.
Koodu ATX: C10AA01

Edemede na-atọ ụtọ

Etu ị ga-esi ahọrọ analọg ziri ezi
Na pharmacology, a na-ekekarị ọgwụ iji mee ka okwu na analogues. Ihe mejuputara ya bu otu uzo ma obu ozo si aru aru nke nwere aru oru aru. Site na analogs bu ogwu eji eme ihe nwere ihe ndi ozo di ndu, mana ebum n’obi iji gwọ oria otu oria a.

Ọdịiche dị n’etiti nje virus na nje
Ọ bụ nje virus, nje, fungi na protozoa na-ebute ọrịa ndị na-efe efe. Ọrịa na-ebute nje na nje na-abụkarị. Agbanyeghị, ịmata ihe kpatara ọrịa ahụ pụtara ịhọrọ usoro ọgwụgwọ dị mma ga-enyere aka ịnagide ọrịa ngwa ngwa na agaghị emerụ nwa ahụ.

Ihe nfụkasị bụ ihe na-akpata otutu oge
Peoplefọdụ ndị maara ọnọdụ nwatakịrị na-arịakarị ụfụ na ogologo oge. Ndị nne na nna na-akpọrọ ya gaa na nke ndị dọkịta, na-ele ule, na-a drugsụ ọgwụ ọjọọ, n'ihi ya, a na-edebanye aha nwatakịrị ahụ na dọkịta ụmụaka mgbe ọ na-arịa ọrịa. Amaghị ihe kpatara ọrịa ọrịa iku ume ugboro ugboro.

Urology: ọgwụgwọ chlamydial urethritis
Chlamydial urethritis na-ahụkarị n’omume urologist. Ọ bụ Chlamidia trachomatis nke nje intracellular, nke nwere akụrụngwa nke nje na nje, nke na-achọkarị ọgwụ mgbochi ogologo oge maka ọgwụgwọ antibacterial. O nwere ike ibute oke urera na ụmụ nwoke na ụmụ nwanyị.

Ariescorp, nkuzi ngwa (usoro na usoro onunu ogwu)

Tupu ịmalite Ovencor ọgwụgwọ, a na-ekenye onye ọrịa ọkọlọtọ nri hypocholesterol. Ọgwụ a ga-a onceụ otu ugboro n'ụbọchị na mgbede, jiri mmiri sachaa ya. Na ntinye nri, ekwesighi ijikọ ọgwụ. Na-atụ aro ọgwụ kwa ụbọchị maka ọgwụgwọ hypercholesterolemia sitere na 10 ruo 80 mg. N'okwu a, ọgwụ izizi bụ 10 mg. A na-eme mgbanwe mgbanwe a na oge nke otu ọnwa. N'ime ọtụtụ ndị ọrịa, ezigbo ọgwụgwọ ọgwụgwọ na-apụta mgbe ị na-ewere Ovenkor na usoro ọgwụ kwa ụbọchị ruo 20 mg.

Maka ndị ọrịa nwere Ọrịa ụbụrụ Ischemic ma ọ bụ nnukwu ihe ọghọm ya nwere ịpụta ọgwụ dị mma kwa ụbọchị bụ ọgwụ 20-40 mg, nke mbido bụ 20 mg kwa ụbọchị. A naghị eme ngagharị dose maka ndị ọrịa mgbe afọ 60 gasị na ndị ọrịa nwere nsogbu ịgbazigharị dị nro ma ọ bụ nke na-adịghị ala. Site na nhazi nke Ovenkoroma na Naerapamil ma obu Amiodarone usoro ubochi nke Ovenkor ekwesịghị ịbụ ihe karịrị 20 mg.

Ngwakọta, ụdị ntọhapụ

Ariescor bụ nkwadebe maka ihe ọkụkụ, yabụ, ọ nwere naanị otu ihe eji eme ihe - simvastatin. Ihe ndị ọzọ fọdụrụnụ na-arụ ọrụ inyeaka: nyejupụta oke, meziwanye mbadamba mbadamba ihe, jikọta ihe niile. N'ime nkwadebe a, a na-eji cellulose, stachi, ascorbic na citric acid, magnesium stearate, titanium dioxide, shuga mmiri ara (lactose), polyethylene glycol 4000, talc na-eji maka ebumnuche ndị a.

Ariescor bụ mbadamba ụrọ nke dị n ’ụzọ abụọ - 10 ma ọ bụ 20 mg. Ha bụ okirikiri, matte, kpuchie ya na shei ọcha.

Omume ọgwụ

A na-ekewa mbadamba nke Ovenkor dị ka prodrugs. Mkpụrụ irighiri simvastatin nwere ọdịdị nke mgbanaka lactone. Dika okwesiri, o nweghi ike iso ndi choro chorol chorol. Ma na imeju, ọ na-arata mgbanwe kemịkal. Simdị simvastatin nọ n'ọrụ yiri nke ahụ na enzyme HMG-CoA reductase, nke dị mkpa maka njikọ cholesterol. N'ihi usoro aghụghọ a, ọ na-ewere ọnọdụ ya na mmeghachi omume kemịkal. Akụkụ ọzọ nke molekul na nke a na - egbochi njikọ cholesterol. Maka nke a, a na-ebelata njikọ nke ihe ndị dị n’ime ya.
Ahụ́ na-eme ka mmiri cholesterol dịkwuo elu site na ịba ụba ọrụ nke ndị na-anabata LDL, na-eme ka mmebi ha dịkwuo ngwa. LDL bụ abụba “jọrọ njọ” nke na-enyere aka itinye nkwụnye ego na mgbidi akwara ọbara. Ya mere, ị Oụ Ovenkor belata ihe ize ndụ nke ịmalite ọrịa atherosclerosis.

Dịka statins ọ bụla, Ovenkor anaghị emetụta ọrụ nke enzymes nke na-akụda abụba (lipases), njikọ, na nkwụsị nke abụba n'efu. Yabụ, mbelata ogo abụba (triglycerides, TG) yikarịrị ka ọ bụ nsonaazụ nke ndị na - anabata mkpụrụ ndụ. Ha na-akpalite mmebi nke mkpụrụ ndụ ihe dị n’etiti dị n’ime ala, 30% mejupụtara TG.

O gosiputara na ojiji nke ogwu Ariescor:

  • na-emetụta steeti nke ala nke arịa ọbara (endothelium), mgbidi nke arịa ọbara,
  • normalizes obara
  • nwere antioxidant Njirimara
  • na-ebelata ọrịa obi.

Dabere na ntuziaka maka Ovenkor, a na-achọpụta ọganihu na steeti endothelium mgbe ọnwa gasịrị.

Ejiri ọgwụ a mara ezigbo mma. Oke itinye uche na ọbara na-aputa na elekere anọ mgbe etinyere mbadamba nke Ovenkor na ahụ. A na-ahụ mgbanwe mbụ dị mma na ọkwa cholesterol mgbe izu abụọ gachara.

Imirikiti simvastatin nwere ihe na-abanye na eriri afọ na-abanye, eriri afọ. Thedị ọgwụ na-adịghị arụ ọrụ nke akụrụ na-ewepụta ya.

Ofzọ nke ngwa, usoro onunu ogwu

Withgwọ ọgwụ na Ovencor chọrọ nri tupu ịmalite ọgwụ, yana oge usoro ọgwụgwọ.

A họrọ ọ̀gwụ nke ọgwụ n’otu n’otu. A na-atụ aro ịmalite iji obere usoro onyonyo, yana mmụba ya. Anyị dere n'elu na a na-enweta mbelata kachasị na cholesterol ụbọchị 28 mgbe mmalite nke ọgwụ. Ọ bụ ya mere mmezi ọgwụ ugboro ugboro anaghị eme uche gị.

Usoro akwadoro ọgwụ nke Ovenkor bụ 5-20 mg / ụbọchị, ihe kachasị bụ 40 mg / ụbọchị. Maka ndị ọrịa na-a immụkwa ọgwụ mgbochi immunosuppressants, iji simvastatin nwere mmachi dị ka 5 mg / ụbọchị. Na nnukwu nsogbu gbasara akụrụ, nkuzi ahụ na-adụ ọdụ site na iji 5-10 mg / ụbọchị.

Nchịkọta ahụ na bioavailability nke ọgwụ ahụ n'ahụ nri adịghị nri. Nwere ike were ya tupu / mgbe nri gasị / mgbe nri, echefula ị notụ nnukwu mmiri. Isi ihe achọrọ dị mkpa: ị kwesịrị ị tabletsụ mbadamba mmanya otu ugboro n'ụbọchị na mgbede.

Mmekorita

Site na nhazi oge nke warfarin na ụfọdụ anticoagulants na Avencor, a na-eme ka mmetụta nke ikpeazụ ahụ ka mma. Ọ na - a potụ mmanya na - egbu egbu nke imeju na - egbu egbu, ọgwụ na - emetụta akụkụ ahụ.

N'ihi ihe ize ndụ nke rhabdomyolysis, ekwenyeghị iji ọgwụ ahụ:

  • ya na keto, itraconazole, otutu nke vitamin PP,
  • ndị mmadụ na-anara ọgwụ mgbochi immunosuppressive.

Ndị dọkịta dere otu okwu banyere mmalite nke rhabdomyolysis mgbe otu ọgwụ simvastatin na sildenafil na-alụ. A na-eji ọgwụ a emezi dysfunction erectile.

Ọnụahịa Ovenkor na-emetụta oke ọnụ ahịa ire ere. N’obodo dị iche iche na ụlọ ahịa ọgwụ Russia, ọ dị ezigbo iche. Ya mere, otu ngwugwu nke 10 mg nwere ike na-eri site na 275 rubles, na usoro 20 mg - site na 419 ruo 578 rubles.

N'ime ụlọ ahịa ọgwụ ọ bụla ị nwere ike ịchọta analogues nke Ovenkor - ọgwụ ọgwụ nwere otu ihe eji arụ ọrụ, mana site na onye nrụpụta dị iche. Simvastatin bụ akụkụ nke: Simvagesal, Zokor, Simvor, Simvakard, Simvastatin, Simvastol, Simgal, Simlo, Vasilip. Na mgbakwunye na ọnụahịa ahụ, ọgwụ ndị a dịgasị iche na usoro dị ọnụ ala. Dịka ọmụmaatụ, enwere ọgwụ nwere 5 na 40 mg nke ihe na-arụ ọrụ. Nke a dabara adaba ma ọ bụrụ na dọkịta ekwuola naanị ụdị ọgwụ a.

Ihe ndi edere n’ere ihe omume a doziri
dị ka usoro nchịkọta akụkọ nke saịtị ahụ si dị.

Ndị na-edoghị anya iji dochie anya Ovenkor

Ihe analogue dị ọnụ ala site na 313 rubles.

Simvastatin bụ ọgwụ Russia nwere oke uru na otu ụdị ihe na-arụ ọrụ na ihe mejupụtara ahụ, mana obere usoro nke 10 mg kwa mbadamba. Edere ya maka ọgwụgwọ nke hypercholesterolemia na hyperlipidemia nke abụọ. Enwere ike ịchọta ndepụta ngosipụta zuru ezu na ntuziaka ahụ.

Simvastol (mbadamba) Rating: 4 Top

Ihe analogue dị ọnụ ala site na 265 rubles.

Simvastol bụ analog nke mmepụta Romania. Odikwa n’ime kaadiboodu nke 14 na mbadamba 28. Ihe na-arụ ọrụ bụ otu ihe ahụ ebe a, yabụ ntuziaka maka ojiji nwere naanị obere ọdịiche. Tupu ịmalite ọgwụgwọ, anyị na-akwadosi ike ịkpọ dọkịta.

Ihe analogue dị ọnụ ala site na 173 rubles.

Ọzọ dochie anya Ovenkor, nke na-enwetakwa uru karịa nke "mbụ", n'agbanyeghị na ọ dịghị iche na ya. Contraindicated na ime, lactation na nwata. Enwere ike ịchọta ndepụta niile nke contraindications na ntuziaka ahụ.

Ahapụ Gị Ikwu